Affinage

RAB8A

Ras-related protein Rab-8A · UniProt P61006

Length
207 aa
Mass
23.7 kDa
Annotated
2026-06-10
100 papers in source corpus 50 papers cited in narrative 51 extracted findings
Cross-family judge vs UniProt: Affinage preferred faithfulness: 6/6 claims corpus-supported (100%)

Mechanistic narrative

Synthesis pass · prose summary of the discoveries below

RAB8A is a prenylated Ras-like small GTPase that operates as a nucleotide-dependent switch governing polarized membrane traffic, cytoskeletal remodeling, and vesicle docking/fusion at the cell surface (PMID:8858170, PMID:9677305). It cycles between an inactive GDP form and an active GTP form set by dedicated regulators: the GEF Rabin8 (GRAB) catalyzes nucleotide exchange with substrate selectivity for RAB8 — a reaction resolved structurally through its ternary GDP, nucleotide-free, and GTP intermediates — and is itself kinetically stimulated by RAB11-GTP enriched at the ciliary base, establishing a RAB11→Rabin8→RAB8A activation cascade (PMID:12221131, PMID:20308558, PMID:24072714). Counterbalancing GAPs including AS160/TBC1D4, the optineurin-recruited TBC1D17, EPI64, the C9ORF72–SMCR8 complex, and the Salmonella effector SopD terminate signaling (PMID:25158853, PMID:22854040, PMID:32303654, PMID:33603205, PMID:22219378). In its GTP-bound state RAB8A engages a panel of effectors — myosin Va/Vb, the autoinhibition-relieving actin-tubulating EHBP1/EHBP1L1–Bin1 module, MICAL3, Slp1/JFC1 and Slp4, and PI3Kγ — to drive cytoskeletal reorganization, exocytic carrier docking and fusion, and effector recruitment to growing membranes (PMID:21596566, PMID:25022365, PMID:24478457, PMID:32826901, PMID:23140275). Through these activities RAB8A controls apical protein delivery and microvillus formation in intestinal epithelia (its loss causing apical mislocalization to lysosomes and microvillus inclusions) (PMID:17597763, PMID:24892806, PMID:26833786), insulin/AMPK-stimulated GLUT4 and CD36 surface translocation downstream of AS160 (PMID:21041651, PMID:22315395, PMID:24478457), primary ciliogenesis via a Rabin8–Sec15 exocyst link (PMID:22433857), LDL-cholesterol recycling and ABCA1-mediated efflux (PMID:24209575, PMID:19304576), lipid-droplet–mitochondria tethering with PLIN5/ATGL in muscle (PMID:36800997), and TLR/LRP1-induced macropinosomal PI3Kγ signaling that tunes inflammatory cytokine output (PMID:25022365, PMID:30208326). LRRK2 phosphorylates RAB8A at Thr72 in switch II, generating a phospho-epitope read by RILPL2 (and JIP3/JIP4) via an X-shaped helical cap that redirects RAB8A to centrosomes and lysosomes; pathogenic LRRK2 mutations exploit this to cause centrosomal cohesion deficits, ciliogenesis defects, and endolysosomal/EGFR trafficking impairment relevant to Parkinson's disease (PMID:29357897, PMID:31428781, PMID:32017888, PMID:30709905).

Mechanistic history

Synthesis pass · year-by-year structured walk · 18 steps
  1. 1993 Medium

    Establishing where RAB8 acts was the first question; peripheral, ruffle-enriched localization distinct from related Rabs defined it as a surface-directed trafficking GTPase.

    Evidence HA-tagged stable expression and immunofluorescence in CHO and Swiss 3T3 cells

    PMID:7688123

    Open questions at the time
    • No functional cargo identified at this stage
    • Single-lab imaging without endogenous validation
  2. 1996 High

    Linking RAB8 activity to outputs showed that active RAB8 reorganizes the cytoskeleton and routes biosynthetic cargo into cell protrusions, tying membrane traffic to cell morphology.

    Evidence Wild-type and Q67L mutant expression with VSV-G trafficking and cytoskeletal imaging in BHK cells; GTP-dependent binding to rab8ip/GC kinase

    PMID:8643544 PMID:8858170

    Open questions at the time
    • rab8ip kinase substrates/function downstream of RAB8 not defined
    • Mechanism coupling RAB8 to actin/microtubules unresolved
  3. 1998 High

    Defining how RAB8 attaches to membranes established it as a CVLL-motif GTPase prenylated predominantly by GGTaseII in a REP-dependent manner.

    Evidence Cell-free prenylation, metabolic mevalonate labeling, and REP-binding-deficient Y78D mutant

    PMID:9677305

    Open questions at the time
    • Does not address regulation of prenylation in vivo
    • Membrane targeting specificity not addressed
  4. 2002 High

    Identifying the activating machinery: Rabin8 was defined as a RAB8-selective GEF that drives cortical actin remodeling and polarized surface domains.

    Evidence Yeast two-hybrid, in vitro GEF assays with substrate selectivity testing, and localization in cells

    PMID:12221131

    Open questions at the time
    • Upstream control of Rabin8 not yet known
    • Effectors mediating actin remodeling unidentified
  5. 2001 High

    In vivo dominant-negative analysis established RAB8 as essential for docking post-Golgi rhodopsin carriers near the ciliary base, the first link to ciliary/photoreceptor traffic.

    Evidence Transgenic Xenopus rod photoreceptors expressing T22N, Q67L, and WT RAB8

    PMID:11514620

    Open questions at the time
    • Docking effectors at the ciliary base not identified
    • Molecular fusion machinery unresolved
  6. 2007 High

    Genetic ablation showed RAB8 is required for apical protein localization in intestinal enterocytes, defining a polarized-trafficking role in vivo.

    Evidence Rab8 knockout mice with immuno-EM and nutrient absorption assays; JRAB/MICAL-L2-mediated E-cadherin transport in epithelia

    PMID:17597763 PMID:18094055

    Open questions at the time
    • Effector machinery for apical sorting not yet defined
    • Compensation by paralogs not addressed at this stage
  7. 2008 Medium

    Connecting RAB8 to metabolic signaling: RAB8A was placed downstream of AS160 with myosin Vb in insulin-stimulated GLUT4 exocytosis.

    Evidence siRNA, dominant-negative myosin Vb fragment, and GLUT4 translocation assays in L6 muscle cells

    PMID:18701652

    Open questions at the time
    • Direct RAB8A-myosin Vb binding not yet shown here
    • GAP identity assumed but not biochemically established at this step
  8. 2010 High

    Defining pathway order in ciliogenesis: RAB11-GTP was shown to directly bind and kinetically stimulate Rabin8, placing RAB11 upstream of the Rabin8–RAB8 axis; insulin-dependent RAB8A GTP loading was placed upstream of RAB13 and downstream of AS160.

    Evidence In vitro GEF kinetics, GST pulldown, RNAi; Rab-GTP activation assays with AS160 epistasis; GPCR C-terminal interaction mapping

    PMID:20308558 PMID:20424170 PMID:21041651

    Open questions at the time
    • Spatial coordination of RAB11/Rabin8/RAB8 cascade not fully resolved
    • How AS160 is inactivated to permit RAB8A loading not detailed
  9. 2011 High

    Dissecting RAB8 in exocytosis and cytokinesis showed it acts at the docking/fusion step (not budding or motility), linked to ELKS via MICAL3, and is delivered to the midbody by DCDC5/dynein.

    Evidence Live-cell vesicle imaging, siRNA, MICAL3 monooxygenase-dead mutant; co-IP and RNAi for DCDC5-dynein

    PMID:21596566 PMID:22159412

    Open questions at the time
    • How MICAL3 monooxygenase remodels the docking complex mechanistically unresolved
    • Coupling of midbody delivery to abscission not detailed
  10. 2012 High

    Mapping the inactivation network: AS160 and EPI64 were defined as RAB8A GAPs, with AS160 controlling lipid-droplet fusion and EPI64 recruiting RAB8A via JFC1; optineurin was shown to scaffold RAB8 with the GAP TBC1D17; Cdc42 was placed upstream of RAB8A activation in epithelia.

    Evidence In vitro GAP assays, ternary complex biochemistry, co-IP, catalytic-dead mutants, lipid droplet/transferrin trafficking readouts, and intestinal conditional knockouts

    PMID:22219378 PMID:22315395 PMID:22354172 PMID:22854040 PMID:25158853

    Open questions at the time
    • Selectivity rules among multiple GAPs not defined
    • How distinct GAPs are spatially targeted to RAB8A pools unresolved
  11. 2013 High

    Expanding effector and physiological scope: RAB8A was shown to mediate cholesterol recycling/efflux with NPC1 and Myosin5b, recruit PI3Kγ via its Ras-binding domain in TLR4 signaling, and use MyoVa as a GTP-selective insulin-responsive effector; the Rabin8-catalyzed exchange reaction was solved structurally.

    Evidence BODIPY-cholesterol imaging, GST pulldown to PI3Kγ RBD, CRISPR/siRNA, MyoVa cargo-tail binding assays, and crystal structures of exchange intermediates

    PMID:23140275 PMID:23175844 PMID:24072714 PMID:24209575 PMID:24478457 PMID:25022365

    Open questions at the time
    • Integration of multiple effectors at a single membrane not resolved
    • How effector choice is determined per pathway unclear
  12. 2013 Medium

    Pre-LRRK2 regulatory mechanism: a GSK3β–Dzip1–GDI2 cascade was shown to control RAB8-GDP release at the ciliary base, and GRAF1-mediated endocytosis was shown to turn over active RAB8 at protrusions, defining spatial control of the RAB8 cycle.

    Evidence In vitro phosphorylation, FRET, basal-body fractionation, shRNA; GRAF1 siRNA with RAB8-GTP measurement and 3D lumen assays

    PMID:25860027 PMID:28137756

    Open questions at the time
    • How GDI extraction is coordinated with GEF activation unresolved
    • Endocytic turnover machinery for active RAB8 incompletely mapped
  13. 2016 High

    Structural and effector mechanism: EHBP1L1–Bin1–dynamin was defined as a RAB8 effector for apical transport, and the EHBP1 bMERB–CH autoinhibition relieved by RAB8 binding explained how RAB8 licenses actin-coupled membrane tubulation.

    Evidence Co-IP, GST pulldown, EHBP1L1 knockout mice; crystal structures of autoinhibited and active EHBP1 states with actin sedimentation

    PMID:24892806 PMID:26833786 PMID:32826901

    Open questions at the time
    • How dynamin scission is timed relative to RAB8 cycling unresolved
    • In vivo requirement of the autoinhibition switch not tested
  14. 2018 High

    Establishing the LRRK2 axis: LRRK2 phosphorylates RAB8A at Thr72 in switch II, redirecting it to centrosomes and causing cohesion/polarity defects reversible by kinase inhibition.

    Evidence In vitro kinase assays, phospho-deficient mutant epistasis, patient-derived cells, and SH-SY5Y stable lines; LRP1-Y4507-dependent RAB8A activation in macropinosomes

    PMID:29357897 PMID:30208326

    Open questions at the time
    • Physiological substrate range of LRRK2 toward RAB8A pools not defined
    • How Thr72 phosphorylation alters the GTPase cycle quantitatively unresolved
  15. 2019 High

    Mechanism of LRRK2 pathology was refined: phospho-RAB8 (with phospho-RAB10) drives RILPL1-dependent centrosomal/ciliary defects and endolysosomal/EGFR trafficking impairment, rescued by the RAB11-Rabin8-RAB8A cascade.

    Evidence Patient-derived and mutant-mouse cells, kinase inhibitor reversal, EGFR trafficking assays with RAB8A variants; oocyte ROCK-LIMK actin study

    PMID:30285101 PMID:30709905 PMID:31428781

    Open questions at the time
    • Why specific compartments accumulate phospho-RAB8 not fully explained
    • Relative contributions of RAB8 vs RAB10 to disease phenotypes unresolved
  16. 2020 High

    Structural recognition of the phospho-switch and inactivation machinery was defined: RILPL2 reads pThr72 via an X-shaped helical cap, and the C9ORF72–SMCR8 complex was shown to be a RAB8A GAP using an arginine-finger mechanism.

    Evidence Crystal structure of phospho-RAB8A·RILPL2 with mutagenesis; cryo-EM of C9ORF72-SMCR8-WDR41 with GAP assays and Arg147 mutagenesis

    PMID:32017888 PMID:32303654

    Open questions at the time
    • Cellular consequences of C9ORF72-SMCR8 GAP activity on RAB8A pools not detailed
    • Generality of phospho-Rab readers beyond RILPL2/JIP3/4 not tested here
  17. 2021 High

    Host–pathogen and lysosomal mistrafficking mechanisms were defined: Salmonella SopD exerts dual GAP/GDI-displacement control over RAB8 to tune inflammation, and gain-of-function LRRK2 sequesters RAB8A to lysosomes, mistrafficking transferrin and altering iron uptake.

    Evidence Crystal structure of SopD-RAB8 with GAP and GDI-displacement assays in infection; LRRK2 kinase inhibitor reversal and iPSC-derived G2019S microglia transferrin assays

    PMID:33603205 PMID:34914695

    Open questions at the time
    • How a single effector achieves opposite activities in vivo not fully resolved
    • Mechanism redirecting RAB8A to lysosomes downstream of phosphorylation incompletely defined
  18. 2023 High

    A non-canonical organelle-tethering role was established: RAB8A serves as a mitochondrial receptor for lipid droplets via PLIN5, recruiting ATGL under AMPK control to couple lipolysis with β-oxidation in muscle.

    Evidence Co-IP, LD-mitochondrion proximity assays, AMPK activation, RAB8A KO mouse exercise phenotype, ATGL recruitment assays

    PMID:36800997

    Open questions at the time
    • How RAB8A switches between vesicle-fusion and tethering functions unresolved
    • Whether GTP-cycle regulators of the tethering role differ from trafficking pools unknown

Open questions

Synthesis pass · forward-looking unresolved questions
  • How a single GTPase selects among its many GAPs, GEFs, and effectors to specify distinct pathways in different cell types remains the central open question.
  • No unified model of spatial/temporal effector selection
  • Quantitative impact of Thr72 phosphorylation on the full GTPase cycle not established
  • Crosstalk between RAB8A trafficking and organelle-tethering functions undefined

Mechanism profile

Synthesis pass · controlled-vocabulary classification · explore literature graph →
Molecular activity
GO:0003924 GTPase activity 7
Localization
GO:0005886 plasma membrane 5 GO:0005929 cilium 4 GO:0005794 Golgi apparatus 3 GO:0005856 cytoskeleton 3 GO:0005764 lysosome 2 GO:0005811 lipid droplet 2 GO:0005815 microtubule organizing center 2
Pathway
R-HSA-9609507 Protein localization 5 R-HSA-1430728 Metabolism 4 R-HSA-1643685 Disease 4 R-HSA-1852241 Organelle biogenesis and maintenance 4 R-HSA-168256 Immune System 3 R-HSA-5653656 Vesicle-mediated transport 3 R-HSA-162582 Signal Transduction 2
Complex memberships
CTLA-4/TRIM/LAX/Rab8 complexEHBP1L1-Bin1-dynamin complexRAB8A-PLIN5 lipid droplet-mitochondrion tethering complex

Evidence

Reading pass · 51 per-paper findings extracted from the source corpus
Year Finding Method Journal Conf PMIDs
1996 Rab8 (wild-type and constitutively active Q67L mutant) expression in BHK fibroblasts promotes reorganization of actin filaments and microtubules, leading to formation of cell protrusions and preferential delivery of newly synthesized basolateral marker protein (VSV-G) into these outgrowths, demonstrating a role for Rab8 in linking polarized biosynthetic membrane traffic to cell morphology changes. Transient expression and stable cell lines with wild-type and mutant Rab8; VSV-G trafficking assay; fluorescence microscopy of actin and microtubule organization The Journal of cell biology High 8858170
1993 Epitope-tagged Rab8, when stably expressed in CHO and Swiss 3T3 cells, localizes to the cell periphery with highest concentration in ruffling areas, distinct from the perinuclear localization of the closely related Rab10, establishing compartment-specific localization for Rab8. HA-epitope tagging, stable transfection, immunofluorescence microscopy Proceedings of the National Academy of Sciences of the United States of America Medium 7688123
1996 Active GTP-bound Rab8 specifically interacts with a murine Rab8-interacting protein (rab8ip/GC kinase), a serine/threonine kinase with autophosphorylation activity, in a GTP-dependent manner; the complex co-immunoprecipitates from transfected cells and both proteins co-localize at the Golgi and basolateral plasma membrane in MDCK cells. Yeast two-hybrid screening, co-immunoprecipitation from transfected 293T cells, cell fractionation, immunofluorescence Proceedings of the National Academy of Sciences of the United States of America Medium 8643544
2000 Active GTP-bound Rab8 interacts with the coiled-coil protein FIP-2, which also binds Huntingtin; co-expression of FIP-2 and Huntingtin enhances recruitment of Huntingtin to Rab8-positive vesicular structures, linking Rab8-mediated membrane trafficking to Huntingtin function. Yeast two-hybrid, co-immunoprecipitation, fluorescence microscopy of co-expressed proteins Current biology : CB Medium 11137014
2001 Dominant-negative Rab8 (T22N) expressed in Xenopus rod photoreceptors causes accumulation of tubulo-vesicular structures at the base of the connecting cilium and rapid retinal degeneration, demonstrating that Rab8 is required for docking of rhodopsin-bearing post-Golgi membranes near the ciliary base. Transgenic Xenopus laevis expressing GFP-tagged wild-type, constitutively active (Q67L), and dominant-negative (T22N) Rab8; fluorescence microscopy; histology Molecular biology of the cell High 11514620
2002 Rabin8 is a Rab8-specific guanine nucleotide exchange factor (GEF) that stimulates nucleotide exchange on Rab8 but not on Rab3A or Rab5; Rabin8 localizes to cortical actin and its expression induces actin remodeling and formation of polarized cell surface domains; dominant-negative Rab8 redistributes Rabin8 from cortical actin to Rab8-specific vesicles. Yeast two-hybrid, in vitro GEF activity assays, fluorescence microscopy, co-expression studies Molecular biology of the cell High 12221131
2006 Endogenous and ectopic Rab8 associates with macropinosomes that form at ruffling membranes; these fuse into tubules recycled to the leading edge; depletion of Rab8 by RNAi inhibits protrusion formation while promoting cell-cell adhesion and stress fibers; Rab8 colocalizes with Rab11 and Arf6, is functionally linked to Arf6, and specifically binds synaptotagmin-like protein Slp1/JFC1. RNAi knockdown, dominant-negative mutant expression, co-localization fluorescence microscopy, binding assays, transferrin trafficking assays Journal of cell science High 17105768
2007 Rab8-knockout mice show mislocalization of apical peptidases and transporters to lysosomes in small intestinal enterocytes, shortened microvilli, enlarged lysosomes, and microvillus inclusions, establishing that Rab8 is required for proper apical protein localization in intestinal epithelial cells. Rab8-deficient mouse knockout, immunofluorescence, electron microscopy, nutrient absorption assays Nature High 17597763
2006 Optineurin interacts with Rab8 and, upon apoptotic stimulus (H2O2), the Rab8 GTPase activity is required for optineurin's translocation from the Golgi to the nucleus; a glaucoma-associated E50K mutant of optineurin loses this ability and compromises mitochondrial membrane integrity. Co-immunoprecipitation, fluorescence microscopy, dominant-negative Rab8, apoptosis assays (cytochrome c release) The Journal of biological chemistry Medium 16569640
2008 Rab8A and myosin Vb are required for insulin-induced GLUT4 translocation in L6 muscle cells; overexpression of a myosin Vb fragment inhibits insulin-stimulated GLUT4 translocation and alters subcellular distribution of GTP-loaded Rab8A, placing them in a common pathway downstream of AS160. siRNA knockdown, overexpression of dominant-negative myosin Vb fragment, GLUT4 translocation assay, immunofluorescence American journal of physiology. Cell physiology Medium 18701652
2007 Rab8 (via JRAB/MICAL-L2) specifically mediates transport of E-cadherin to the plasma membrane independently of Rab13; Rab8 and Rab13 compete for binding to JRAB/MICAL-L2 and associate with it at different compartments (perinuclear recycling/storage and plasma membrane respectively) to coordinate AJ and TJ assembly. siRNA knockdown, co-immunoprecipitation, Ca²⁺-switch model, fluorescence microscopy Molecular biology of the cell Medium 18094055
2010 Rab11-GTP binds directly to Rabin8 and kinetically stimulates its GEF activity toward Rab8; Rab11 enriches at the base of primary cilia and dominant-negative Rab11 or RNAi of Rab11 blocks ciliogenesis, placing Rab11 upstream of Rabin8-Rab8 in a vesicular trafficking cascade required for primary ciliogenesis. GEF kinetic assays in vitro, GST pulldown, dominant-negative expression, RNAi, immunofluorescence microscopy Proceedings of the National Academy of Sciences of the United States of America High 20308558
2010 Insulin promotes GTP loading of Rab8A in rat L6 muscle cells; Rab8A is activated upstream of Rab13 in response to insulin; both Rab8A and Rab13 are targets of the AS160 GAP activity, and overexpression of Rab8A or Rab13 reverses constitutively active AS160-mediated suppression of surface GLUT4. Rab-GTP pull-down activation assay, siRNA knockdown, constitutively active AS160 overexpression, surface GLUT4 quantification Proceedings of the National Academy of Sciences of the United States of America High 21041651
2011 Rab8A stably associates with exocytotic vesicles in a Rab6-dependent manner; Rab8A function is required for docking and fusion of exocytotic carriers but not for their budding or motility; Rab8A and ELKS act in the same pathway linked by MICAL3, whose monooxygenase activity is required for vesicle-docking complex remodeling. Live-cell imaging of vesicle dynamics, siRNA knockdown, co-localization, dominant-negative constructs, MICAL3 monooxygenase-dead mutant Current biology : CB High 21596566
2012 Rabin8 interacts with Sec15 (exocyst subunit) in a conformation-dependent manner enhanced by constitutively active Rab8; Sec15 co-localizes with Rab8 along the primary cilium; inhibition of Sec15 causes ciliogenesis defects, establishing a Rabin8-Rab8-Sec15 interaction that couples Rab8 activation to effector recruitment for ciliary vesicle trafficking. Co-immunoprecipitation, immunofluorescence microscopy, constitutively active Rab8 expression, Sec15 siRNA knockdown, ciliogenesis assay The Journal of biological chemistry High 22433857
2012 Cdc42 deficiency impairs Rab8a activation and its association with multiple effectors, and prevents Rab8a vesicle trafficking to the midbody, impeding cytokinesis; Rab8a is also required for Cdc42-GTP activity in intestinal epithelium, and haploinsufficiency of both Cdc42 and Rab8a causes abnormal crypt morphogenesis. Conditional intestinal epithelium-specific knockout mice, immunofluorescence, Rab8a activation assays, genetic interaction (double haploinsufficiency) The Journal of clinical investigation High 22354172
2012 AS160 is the GTPase-activating protein (GAP) for Rab8a; AS160 forms a ternary complex with Fsp27 and Rab8a; GDP-bound Rab8a (inactivated by AS160) promotes lipid droplet fusion; MSS4 (a GEF) antagonizes this activity through Rab8a, establishing an AS160-Rab8a-MSS4 regulatory circuit controlling lipid droplet fusion. In vitro GAP activity assays, co-immunoprecipitation, pulldown, lipid droplet fusion assays in adipocytes, siRNA knockdown in ob/ob mouse livers Developmental cell High 25158853
2012 AS160 mediates insulin- and AMPK-stimulated surface translocation of CD36 in cardiomyocytes; Rab8a GTPase specifically mediates CD36 membrane recruitment upon insulin/AICAR stimulation, established by overexpression and knockdown studies. AS160 overexpression and siRNA knockdown, Rab8a overexpression and knockdown, surface CD36 quantification by immunofluorescence and flow cytometry Journal of lipid research Medium 22315395
2012 Optineurin acts as an adaptor to bring together Rab8 and its GAP TBC1D17; TBC1D17 catalytic activity inhibits Rab8-mediated endocytic recycling of transferrin receptor by preventing Rab8 recruitment to endocytic recycling tubules; the glaucoma-associated E50K optineurin mutant causes enhanced inhibition of Rab8 by TBC1D17. Co-immunoprecipitation, siRNA knockdown, dominant-negative and catalytic-dead mutants, fluorescence microscopy of transferrin receptor trafficking Journal of cell science High 22854040
2013 Rab8a-knockout mice (single and double with Rab8b) show mislocalization of apical markers to lysosomes; Rab8a and Rab8b have compensatory roles in apical transport but do not significantly affect basolateral/dendritic transport; additional knockdown of Rab10 in double-KO cells greatly reduces ciliated cells, indicating Rab8a/b and Rab10 cooperate for ciliogenesis. Single and double knockout mice, immunofluorescence, electron microscopy, Rab10 siRNA in double-KO cells, ciliation quantification Journal of cell science High 24213529
2013 Rab8A directly interacts with PI3Kγ through PI3Kγ's Ras-binding domain; Rab8a recruits PI3Kγ to LPS-induced dorsal ruffles on macrophages to regulate Akt/mTOR signaling downstream of surface TLR4, biasing cytokine output to suppress inflammation. Co-immunoprecipitation, GST pulldown with PI3Kγ Ras-binding domain, CRISPR/siRNA knockdown, cytokine measurement, phospho-Akt assays Nature communications High 25022365
2013 Rab8a regulates LDL cholesterol recycling to the plasma membrane: NPC1 is required to recruit Rab8a to cholesterol-containing late endosomes; Rab8a and Myosin5b cooperate to dock cholesterol-containing carriers to cortical actin near focal adhesions; Rab8a-dependent cholesterol delivery stimulates cell migration. BODIPY-cholesterol live cell imaging, siRNA knockdown of Rab8a/NPC1/Myo5b, immunofluorescence, migration assays Developmental cell High 24209575
2013 Structural snapshots of the complete nucleotide exchange reaction of Rab8 catalyzed by Rabin8/GRAB were obtained, including ternary Rab8·GEF·GDP, binary nucleotide-free Rab8·GEF, and ternary Rab8·GEF·GTP complexes, providing mechanistic detail of GEF-catalyzed nucleotide exchange. X-ray crystallography and enzymatic kinetic characterization of exchange intermediates The Journal of biological chemistry High 24072714
2014 MyoVa is an effector of Rab8A in insulin-stimulated GLUT4 vesicle exocytosis in muscle cells; the MyoVa cargo-binding C-terminal tail binds preferentially to GTP-locked Rab8A in an insulin- and PI3K-dependent manner; MyoVa-CT overexpression and MyoVa siRNA both inhibit insulin-stimulated GLUT4 surface translocation. GST pulldown assays, co-localization fluorescence microscopy, TIRF microscopy, siRNA knockdown, dominant-negative MyoVa-CT overexpression Molecular biology of the cell High 24478457
2014 MYO5B (myosin Vb) uncoupling from RAB8A (and RAB11A) elicits microvillus inclusion disease phenotype; microvilli establishment requires interaction between RAB8A and MYO5B; loss of RAB8A–MYO5B interaction leads to loss of microvilli while loss of RAB11A–MYO5B interaction induces microvillus inclusions. Stable MYO5B knockdown in CaCo2-BBE cells, expression of MVID-associated MYO5B-P660L mutant, surface biotinylation, dual immunofluorescence The Journal of clinical investigation High 24892806
2015 Rab8a mediates anterograde transport of Gpr177 (wntless, the Wnt-specific transporter); Gpr177 binds Rab8a, and depletion of Rab8a compromises Gpr177 trafficking and Wnt secretion, reducing Wnt/β-catenin signaling, severely impairing Paneth cell maturation, and decreasing plasma membrane localization of Gpr177. Co-immunoprecipitation, Rab8a knockout mouse intestinal organoids, immunogold electron microscopy, surface protein biotinylation, Wnt signaling reporter assays Development (Cambridge, England) High 26015543
2015 GSK3β phosphorylates Dzip1 at S520 in G0 phase, increasing Dzip1 binding to GDI2 and promoting release of Rab8-GDP at the cilium base; Dzip1 preferentially binds Rab8-GDP and promotes its dissociation from GDI2 at the pericentriolar region; loss of Dzip1 causes failed ciliary localization of Rab8, establishing a GSK3β-Dzip1-Rab8 cascade regulating post-mitotic ciliogenesis. In vitro phosphorylation assay, FRET, immunoprecipitation, sucrose gradient centrifugation of basal bodies, mass spectrometry phosphopeptide identification, GST pulldown, shRNA knockdown PLoS biology High 25860027
1998 Rab8, which ends in a CVLL motif, can be prenylated by either GGTaseII (REP-dependent) or GGTaseI (REP-independent) in cell-free assays; in vivo labeling experiments show GGTaseII is the predominant enzyme for Rab8 prenylation in human cells, as a REP-binding-deficient Rab8 Y78D mutant shows ~60-70% reduced prenylation. Cell-free prenylation assays, metabolic [³H]mevalonate labeling, GGTaseI inhibitor GGTI-298 treatment, REP-binding-deficient mutant Y78D The Biochemical journal High 9677305
2016 EHBP1L1 directly binds GTP-loaded Rab8 and Bin1; EHBP1L1-Bin1-dynamin complex at the endocytic recycling compartment is required for apical (but not basolateral) protein transport; EHBP1L1-deficient mice show truncated microvilli in small intestine, establishing EHBP1L1 as a Rab8 effector for apical transport. Co-immunoprecipitation, GST pulldown, knockdown in intestinal organoids, EHBP1L1 knockout mice, immunofluorescence The Journal of cell biology High 26833786
2016 GRAF1-mediated clathrin-independent endocytosis removes active Rab8 from the plasma membrane at protrusions; GRAF1 depletion leads to elevated GTP-loaded Rab8 accumulated at static protrusion tips and impairs multi-directional spreading and 3D lumen formation, indicating that endocytic turnover of Rab8 controls cell polarization. GRAF1 siRNA knockdown, Rab8-GTP level measurement, live-cell imaging, 3D culture lumen assay Journal of cell science Medium 28137756
2018 LRRK2 phosphorylates Rab8a at T72 in its switch II domain; pathogenic LRRK2 mutations increase centrosomal localization of phospho-Rab8a, causing centrosomal cohesion deficits and polarity defects; these defects are mimicked by co-expression of wild-type LRRK2 with wild-type but not phospho-deficient Rab8a, and are reversed by LRRK2 kinase inhibition or Rab8a RNAi. In vitro kinase assays, co-immunoprecipitation, GTP binding/retention assays, immunofluorescence, siRNA, patient-derived peripheral cells, SH-SY5Y stable cell lines Molecular neurodegeneration High 29357897
2018 TLR activation of LRP1 results in LRP1 phosphorylation at Y4507, which allows LRP1 to activate and recruit Rab8a together with the PI3Kγ p110γ/p101 effector complex on macropinosomal membranes; in LRP1-deficient cells, TLR-induced Rab8a activation is abolished, altering Akt/mTOR signaling and producing a pro-inflammatory cytokine bias. CRISPR knockout of LRP1, co-immunoprecipitation, phospho-LRP1 analysis, Rab8a activation assay, cytokine measurement Cell reports High 30208326
2019 Pathogenic LRRK2 G2019S expression or loss of RAB8A both impair endolysosomal trafficking and EGFR degradation, causing EGFR accumulation in a RAB4-positive compartment with deficits in recycling; up-regulation of the RAB11-Rabin8-RAB8A cascade or expression of active/phosphodeficient RAB8A variants rescue G2019S LRRK2-mediated trafficking defects, placing RAB8A downstream of LRRK2 in endolysosomal regulation. Immunofluorescence, pulldown assays, RAB8A siRNA knockdown, dominant-negative and constitutively active RAB8A variants, EGFR trafficking assay The Journal of biological chemistry Medium 30709905
2019 RAB8 and RAB10 both contribute to LRRK2-mediated centrosomal cohesion deficits and ciliogenesis defects; pathogenic LRRK2 causes centrosomal accumulation of both phospho-RAB8 and phospho-RAB10, and both effects are dependent on RILPL1; these defects are observed in patient-derived peripheral cells and primary astrocytes from mutant LRRK2 mice. Immunofluorescence in patient-derived cells, primary LRRK2 mouse astrocytes, LRRK2 kinase inhibitor treatment, phospho-RAB8/RAB10 detection Human molecular genetics High 31428781
2020 Crystal structure of phospho-Rab8a (pT72) in complex with the RH2 domain of RILPL2 reveals a heterotetramer where RILPL2 forms an X-shaped α-helical dimer bridging two pRab8a molecules; conserved Arg residues in the RILPL2 X-cap orient toward pT72; similar X-cap residues in JIP3 and JIP4 also interact with LRRK2-phosphorylated Rabs, defining a general recognition mode for phospho-Rab GTPases. X-ray crystallography, structure-function mutagenesis, biochemical binding assays Structure (London, England : 1993) High 32017888
2020 Cryo-EM structure of the C9ORF72-SMCR8-WDR41 complex shows that SMCR8 Arg147 acts as an arginine finger analogous to FLCN, and biochemical assays demonstrate GAP activity of the C9ORF72-SMCR8 complex toward Rab8a and Rab11a. Cryo-EM structure at 3.2 Å, biochemical GAP activity assays, Arg147 mutagenesis Proceedings of the National Academy of Sciences of the United States of America High 32303654
2020 The bMERB domain of EHBP1 forms an intramolecular auto-inhibitory complex with the central calponin homology (CH) domain, preventing actin binding; Rab8 family member binding to bMERB relieves this inhibition and frees the CH domain to interact with actin, promoting membrane tubulation. Crystal structures of the auto-inhibited CH:bMERB and active bMERB:Rab8 complexes were determined. X-ray crystallography, biochemical binding assays, actin sedimentation assays, structure-based mutagenesis Nature communications High 32826901
2021 Salmonella effector SopD has GAP activity for Rab8 (inhibiting Rab8 and stimulating inflammation) and also activates Rab8 by displacing it from its GDI (suppressing inflammation); the crystal structure of SopD bound to Rab8 at 2.3 Å reveals a unique contact interface underlying these dual activities. GAP activity assay, GDI displacement assay, crystal structure at 2.3 Å, Salmonella infection models Nature microbiology High 33603205
2021 LRRK2 gain-of-function mutations induce sequestration of Rab8a to lysosomes in cells; pharmacological inhibition of LRRK2 kinase activity reverses this lysosomal sequestration; LRRK2 mutations drive co-association of endocytosed transferrin with Rab8a-positive lysosomes, and iPSC-derived microglia from LRRK2 G2019S patients mistraffic transferrin to lysosomes, altering iron uptake. LRRK2 kinase inhibitor treatment, immunofluorescence, transferrin trafficking assay, iPSC-derived microglia, G2019S knock-in mice with LPS challenge PLoS biology Medium 34914695
2023 Rab8a acts as a mitochondrial receptor for lipid droplets in skeletal muscle, forming a tethering complex with LD-associated PLIN5; AMPK increases GTP-bound Rab8a upon starvation, promoting LD-mitochondrion interaction; the Rab8a-PLIN5 complex recruits ATGL to couple fatty acid mobilization from LDs with mitochondrial β-oxidation; Rab8a deficiency impairs fatty acid utilization and decreases exercise endurance in mice. Co-immunoprecipitation, LD-mitochondrion proximity assay, AMPK activation, Rab8a KO mouse exercise model, ATGL recruitment assay Developmental cell High 36800997
2010 Rab8 interacts with distinct motifs in the C-termini of α2B- and β2-adrenergic receptors via GST pulldown and co-immunoprecipitation; GDP-bound Rab8(T22N) arrests α2B-AR but not β2-AR in the trans-Golgi network and attenuates ERK1/2 activation by α2B-AR; knockdown of Rab8 more potently inhibits α2B-AR cell surface expression. Co-immunoprecipitation, GST fusion protein pulldown, dominant-negative Rab8, shRNA knockdown, ERK1/2 activation assay, receptor surface expression quantification The Journal of biological chemistry Medium 20424170
2012 Optineurin mediates the interaction between Rab8 and TBC1D17 (a RabGAP); a non-catalytic region of TBC1D17 interacts directly with optineurin; through catalytic activity, TBC1D17 inhibits Rab8 recruitment to endocytic recycling tubules and impairs transferrin receptor recycling; a glaucoma-associated optineurin mutant E50K causes enhanced inhibition of Rab8 by TBC1D17. Co-immunoprecipitation, GST pulldown, siRNA knockdown, dominant-negative constructs, transferrin receptor trafficking assay, fluorescence microscopy Journal of cell science High 22854040
2011 DCDC5 interacts with cytoplasmic dynein, Rab8, and Rabin8; DCDC5 knockdown impairs entry of Golgi-derived Rab8-positive vesicles to the midbody and increases multinucleated cells, demonstrating that DCDC5 mediates dynein-dependent transport of Rab8-positive vesicles during cytokinesis. Co-immunoprecipitation, RNAi knockdown, live-cell imaging of Rab8 vesicles, mitosis/cytokinesis quantification Journal of cell science Medium 22159412
2014 LAX binds active GTP-bound Rab8 via its N-terminus and also binds the cytoplasmic tail of CTLA-4; TRIM requires LAX for Rab8 binding; together they form a CTLA-4/TRIM/LAX/Rab8 complex; disruption of LAX/Rab8 binding reduces CTLA-4-containing vesicle numbers near the TGN and decreases CTLA-4 surface expression on T cells. Co-immunoprecipitation, siRNA knockdown of LAX and Rab8, surface CTLA-4 quantification, vesicle counting by fluorescence microscopy Molecular and cellular biology Medium 24515439
2016 Rab8 activation induces Rac1/Tiam1-mediated cortical actin polymerization and RhoA-dependent stress fiber disassembly; Rab8 promotes focal adhesion disassembly in a microtubule-, calpain-, and MT1-MMP-dependent manner; Rab8 is required for EGF-induced cell polarization and chemotaxis. High-content fluorescence microscopy analysis, Rac1/RhoA activity assays, Rab8 depletion/activation, inhibitor studies (calpain, MT1-MMP), chemotaxis assays Journal of cell science Medium 26940916
2017 TMEM230 depletion inhibits Rab8a-mediated secretory vesicle trafficking, impairs extracellular secretion of p62 and lysosomal hydrolases, disrupts retromer cargo CI-M6PR trafficking, and impairs autophagic cargo degradation; LRRK2 knockdown similarly impairs these Rab8a-dependent functions. siRNA knockdown of TMEM230 and LRRK2, secretion assays, immunofluorescence, retromer localization Human molecular genetics Medium 28115417
2019 RAB8A GTPase localizes to the spindle periphery and cortex in mouse oocytes; RAB8A depletion decreases cytoplasmic and cortical actin filaments, causing spindle migration defects, polar body extrusion failure, and Golgi distribution disruption; RAB8A promotes actin assembly through the ROCK-LIMK signaling pathway and interacts with Golgi marker GM130. Confocal microscopy, RAB8A morpholino/siRNA depletion, mass spectrometry, co-immunoprecipitation with GM130, ROCK inhibitor, actin quantification Biology of reproduction Medium 30285101
2009 Rab8 depletion in primary human macrophages decreases the fraction of ABCA1 at the plasma membrane and inhibits efflux of lipoprotein-derived endosomal cholesterol to apoA-I; Rab8 overexpression increases ABCA1 protein levels and reduces cholesterol deposition, establishing Rab8 as a regulator of ABCA1 surface delivery and cholesterol efflux. Adenoviral overexpression, siRNA knockdown, ABCA1 surface localization quantification, cholesterol efflux assay to apoA-I Arteriosclerosis, thrombosis, and vascular biology Medium 19304576
2012 EPI64's RabGAP domain has GAP activity toward Rab8a; EPI64 binds JFC1 (Slp1, an effector of Rab8a-GTP) via its C-terminal region; EPI64 expression lowers Rab8-GTP levels and coexpression of Rab8a suppresses EPI64-induced vacuole formation, suggesting that EPI64 recruits Rab8a-GTP via JFC1 for deactivation. Co-localization, co-immunoprecipitation, Rab8-GTP level assay, mutant EPI64 lacking GAP activity, Rab8a co-expression rescue Molecular biology of the cell Medium 22219378
2013 Rab8 interacts with the C-terminal tail of mGluR1a in an agonist-dependent manner; Rab8 expression attenuates mGluR1a-mediated inositol phosphate formation and calcium release in a PKC-dependent manner while increasing mGluR1a cell surface expression by decreasing receptor endocytosis. Co-immunoprecipitation, dominant-negative/constitutively active Rab8, inositol phosphate assay, calcium imaging, surface receptor quantification The Journal of neuroscience : the official journal of the Society for Neuroscience Medium 23175844
2013 Slp4 interacts with Rab8 preferentially in its GTP-bound form via the Slp-homology domain; Slp4 and Rab8 colocalize at the plasma membrane in transfected cells and in the center of activated platelets; both Slp4 and Rab8 enhance dense granule release and the Slp4 effect is dependent on Rab8 binding. GST pulldown, co-immunoprecipitation, live microscopy, permeabilized platelet secretion assay Journal of thrombosis and haemostasis : JTH Medium 23140275

Source papers

Stage 0 corpus · 100 papers · ranked by NIH iCite citations
Year Title Journal Citations PMID
2010 Coordination of Rab8 and Rab11 in primary ciliogenesis. Proceedings of the National Academy of Sciences of the United States of America 402 20308558
2003 The BTB protein MEL-26 is a substrate-specific adaptor of the CUL-3 ubiquitin-ligase. Nature 361 13679921
2007 The Rab8 GTPase regulates apical protein localization in intestinal cells. Nature 284 17597763
1996 Rab8 promotes polarized membrane transport through reorganization of actin and microtubules in fibroblasts. The Journal of cell biology 222 8858170
2001 Mutant rab8 Impairs docking and fusion of rhodopsin-bearing post-Golgi membranes and causes cell death of transgenic Xenopus rods. Molecular biology of the cell 206 11514620
1999 The role of CD146 (Mel-CAM) in biology and pathology. The Journal of pathology 202 10451481
2003 Targeted disruption of the mouse Mel(1b) melatonin receptor. Molecular and cellular biology 193 12529409
2006 Characterization of the Rab8-specific membrane traffic route linked to protrusion formation. Journal of cell science 186 17105768
2000 FIP-2, a coiled-coil protein, links Huntingtin to Rab8 and modulates cellular morphogenesis. Current biology : CB 183 11137014
2002 A Rab8-specific GDP/GTP exchange factor is involved in actin remodeling and polarized membrane transport. Molecular biology of the cell 175 12221131
2011 Rab6, Rab8, and MICAL3 cooperate in controlling docking and fusion of exocytotic carriers. Current biology : CB 163 21596566
2010 Rab8A and Rab13 are activated by insulin and regulate GLUT4 translocation in muscle cells. Proceedings of the National Academy of Sciences of the United States of America 148 21041651
1993 Expression and localization of two low molecular weight GTP-binding proteins, Rab8 and Rab10, by epitope tag. Proceedings of the National Academy of Sciences of the United States of America 142 7688123
2012 A Rab8 guanine nucleotide exchange factor-effector interaction network regulates primary ciliogenesis. The Journal of biological chemistry 118 22433857
2006 MEL-28, a novel nuclear-envelope and kinetochore protein essential for zygotic nuclear-envelope assembly in C. elegans. Current biology : CB 115 16950114
2008 Muscle cells engage Rab8A and myosin Vb in insulin-dependent GLUT4 translocation. American journal of physiology. Cell physiology 114 18701652
2014 Rab8a interacts directly with PI3Kγ to modulate TLR4-driven PI3K and mTOR signalling. Nature communications 111 25022365
2006 Optineurin increases cell survival and translocates to the nucleus in a Rab8-dependent manner upon an apoptotic stimulus. The Journal of biological chemistry 109 16569640
2013 Rab8a and Rab8b are essential for several apical transport pathways but insufficient for ciliogenesis. Journal of cell science 108 24213529
2012 The Arf GAP ASAP1 provides a platform to regulate Arf4- and Rab11-Rab8-mediated ciliary receptor targeting. The EMBO journal 107 22983554
2014 Rab8a-AS160-MSS4 regulatory circuit controls lipid droplet fusion and growth. Developmental cell 106 25158853
2007 The interaction of JRAB/MICAL-L2 with Rab8 and Rab13 coordinates the assembly of tight junctions and adherens junctions. Molecular biology of the cell 102 18094055
2012 Insulin and AMPK regulate FA translocase/CD36 plasma membrane recruitment in cardiomyocytes via Rab GAP AS160 and Rab8a Rab GTPase. Journal of lipid research 100 22315395
2002 Rho-binding kinase (LET-502) and myosin phosphatase (MEL-11) regulate cytokinesis in the early Caenorhabditis elegans embryo. Journal of cell science 98 12006612
2010 BMI1 and Mel-18 oppositely regulate carcinogenesis and progression of gastric cancer. Molecular cancer 97 20170541
2013 LDL cholesterol recycles to the plasma membrane via a Rab8a-Myosin5b-actin-dependent membrane transport route. Developmental cell 96 24209575
2012 Cdc42 and Rab8a are critical for intestinal stem cell division, survival, and differentiation in mice. The Journal of clinical investigation 93 22354172
2014 Myosin Vb uncoupling from RAB8A and RAB11A elicits microvillus inclusion disease. The Journal of clinical investigation 91 24892806
1999 Tight association of the human Mel(1a)-melatonin receptor and G(i): precoupling and constitutive activity. Molecular pharmacology 91 10531408
1996 In its active form, the GTP-binding protein rab8 interacts with a stress-activated protein kinase. Proceedings of the National Academy of Sciences of the United States of America 90 8643544
2011 Rab8 GTPase as a regulator of cell shape. Cytoskeleton (Hoboken, N.J.) 86 21850707
2023 Rab8a as a mitochondrial receptor for lipid droplets in skeletal muscle. Developmental cell 85 36800997
2010 Melatonin decreases cell proliferation and induces melanogenesis in human melanoma SK-MEL-1 cells. Journal of pineal research 85 20459460
1997 Melanoma cell-cell interactions are mediated through heterophilic Mel-CAM/ligand adhesion. Cancer research 85 9288796
2018 Parkinson disease-associated mutations in LRRK2 cause centrosomal defects via Rab8a phosphorylation. Molecular neurodegeneration 81 29357897
1997 The cell-cell adhesion receptor Mel-CAM acts as a tumor suppressor in breast carcinoma. The American journal of pathology 78 9284823
2019 RAB8, RAB10 and RILPL1 contribute to both LRRK2 kinase-mediated centrosomal cohesion and ciliogenesis deficits. Human molecular genetics 74 31428781
2021 Mutations in LRRK2 linked to Parkinson disease sequester Rab8a to damaged lysosomes and regulate transferrin-mediated iron uptake in microglia. PLoS biology 72 34914695
2018 TLR Crosstalk Activates LRP1 to Recruit Rab8a and PI3Kγ for Suppression of Inflammatory Responses. Cell reports 72 30208326
2014 Myosin Va mediates Rab8A-regulated GLUT4 vesicle exocytosis in insulin-stimulated muscle cells. Molecular biology of the cell 72 24478457
2019 Antiproliferative and apoptotic effects of caffeic acid on SK-Mel-28 human melanoma cancer cells. Molecular biology reports 71 30719606
2015 The Ciliopathy Protein CC2D2A Associates with NINL and Functions in RAB8-MICAL3-Regulated Vesicle Trafficking. PLoS genetics 71 26485645
2015 Rab8, POSH, and TAK1 regulate synaptic growth in a Drosophila model of frontotemporal dementia. The Journal of cell biology 68 25800055
2020 LRRK2 Is Recruited to Phagosomes and Co-recruits RAB8 and RAB10 in Human Pluripotent Stem Cell-Derived Macrophages. Stem cell reports 65 32359446
2020 Structural Basis for Rab8a Recruitment of RILPL2 via LRRK2 Phosphorylation of Switch 2. Structure (London, England : 1993) 64 32017888
2020 Cryo-EM structure of C9ORF72-SMCR8-WDR41 reveals the role as a GAP for Rab8a and Rab11a. Proceedings of the National Academy of Sciences of the United States of America 61 32303654
2019 The G2019S variant of leucine-rich repeat kinase 2 (LRRK2) alters endolysosomal trafficking by impairing the function of the GTPase RAB8A. The Journal of biological chemistry 60 30709905
2012 Optineurin mediates a negative regulation of Rab8 by the GTPase-activating protein TBC1D17. Journal of cell science 57 22854040
2006 Biosurfactant MEL-A enhances cellular association and gene transfection by cationic liposome. Journal of controlled release : official journal of the Controlled Release Society 57 16624437
2017 Small GTPase Rab8a-recruited Phosphatidylinositol 3-Kinase γ Regulates Signaling and Cytokine Outputs from Endosomal Toll-like Receptors. The Journal of biological chemistry 56 28130450
1998 mel-18 negatively regulates cell cycle progression upon B cell antigen receptor stimulation through a cascade leading to c-myc/cdc25. Immunity 56 9806630
2016 C9ORF72 is a GDP/GTP exchange factor for Rab8 and Rab39 and regulates autophagy. Small GTPases 55 27494456
2013 Intermediates in the guanine nucleotide exchange reaction of Rab8 protein catalyzed by guanine nucleotide exchange factors Rabin8 and GRAB. The Journal of biological chemistry 55 24072714
2016 EHBP1L1 coordinates Rab8 and Bin1 to regulate apical-directed transport in polarized epithelial cells. The Journal of cell biology 53 26833786
2016 Protease-Resistant and Cell-Permeable Double-Stapled Peptides Targeting the Rab8a GTPase. ACS chemical biology 52 27336832
2010 Rab8 interacts with distinct motifs in alpha2B- and beta2-adrenergic receptors and differentially modulates their transport. The Journal of biological chemistry 52 20424170
2013 The PCP effector Fuzzy controls cilial assembly and signaling by recruiting Rab8 and Dishevelled to the primary cilium. Molecular biology of the cell 51 23303251
2001 Ceramide inhibits cell proliferation through Akt/PKB inactivation and decreases melanin synthesis in Mel-Ab cells. Pigment cell research 50 11310790
2017 The Parkinson's disease-linked protein TMEM230 is required for Rab8a-mediated secretory vesicle trafficking and retromer trafficking. Human molecular genetics 48 28115417
2015 GSK3β-Dzip1-Rab8 cascade regulates ciliogenesis after mitosis. PLoS biology 48 25860027
2015 Rab8a vesicles regulate Wnt ligand delivery and Paneth cell maturation at the intestinal stem cell niche. Development (Cambridge, England) 46 26015543
2017 Abnormal Rab11-Rab8-vesicles cluster in enterocytes of patients with microvillus inclusion disease. Traffic (Copenhagen, Denmark) 44 28407399
2020 Synergistic antibacterial and antibiofilm effects of ultrasound and MEL-A against methicillin-resistant Staphylococcus aureus. Ultrasonics sonochemistry 43 33388695
2018 Rab11a-Rab8a cascade regulates the formation of tunneling nanotubes through vesicle recycling. Journal of cell science 41 30209134
2016 Identification of Conserved MEL-28/ELYS Domains with Essential Roles in Nuclear Assembly and Chromosome Segregation. PLoS genetics 41 27341616
2021 AGC kinases and MAB4/MEL proteins maintain PIN polarity by limiting lateral diffusion in plant cells. Current biology : CB 40 33705718
2012 Rab8a regulates the exocyst-mediated kiss-and-run discharge of the Dictyostelium contractile vacuole. Molecular biology of the cell 40 22323285
2011 Linking cytoplasmic dynein and transport of Rab8 vesicles to the midbody during cytokinesis by the doublecortin domain-containing 5 protein. Journal of cell science 38 22159412
2009 Rab8 regulates ABCA1 cell surface expression and facilitates cholesterol efflux in primary human macrophages. Arteriosclerosis, thrombosis, and vascular biology 38 19304576
2008 Rab8-optineurin-myosin VI: analysis of interactions and functions in the secretory pathway. Methods in enzymology 38 18413238
1998 Prenylation of Rab8 GTPase by type I and type II geranylgeranyl transferases. The Biochemical journal 38 9677305
2018 LRRK2 mediated Rab8a phosphorylation promotes lipid storage. Lipids in health and disease 37 29482628
2001 Ovarian expression of melatonin Mel(1a) receptor mRNA during mouse development. Molecular reproduction and development 36 11389547
2021 The Salmonella effector protein SopD targets Rab8 to positively and negatively modulate the inflammatory response. Nature microbiology 35 33603205
2012 Rab8 modulates metabotropic glutamate receptor subtype 1 intracellular trafficking and signaling in a protein kinase C-dependent manner. The Journal of neuroscience : the official journal of the Society for Neuroscience 33 23175844
2020 GRAF2, WDR44, and MICAL1 mediate Rab8/10/11-dependent export of E-cadherin, MMP14, and CFTR ΔF508. The Journal of cell biology 32 32344433
2014 Dihydromyricetin induces cell cycle arrest and apoptosis in melanoma SK-MEL-28 cells. Oncology reports 32 24789439
2016 Small GTPases Rab8a and Rab11a Are Dispensable for Rhodopsin Transport in Mouse Photoreceptors. PloS one 31 27529348
2015 MEL-18 loss mediates estrogen receptor-α downregulation and hormone independence. The Journal of clinical investigation 30 25822021
2011 RAB8 enhances TMEM205-mediated cisplatin resistance. Pharmaceutical research 30 21969054
2010 Protein kinase WNK1 promotes cell surface expression of glucose transporter GLUT1 by regulating a Tre-2/USP6-BUB2-Cdc16 domain family member 4 (TBC1D4)-Rab8A complex. The Journal of biological chemistry 29 20937822
2020 The mechanism of activation of the actin binding protein EHBP1 by Rab8 family members. Nature communications 28 32826901
2016 Rab8 directs furrow ingression and membrane addition during epithelial formation in Drosophila melanogaster. Development (Cambridge, England) 28 26839362
2013 Synaptotagmin-like protein 4 and Rab8 interact and increase dense granule release in platelets. Journal of thrombosis and haemostasis : JTH 28 23140275
1996 Diagnostic and biological implications of mel-CAM expression in mesenchymal neoplasms. Clinical cancer research : an official journal of the American Association for Cancer Research 28 9816205
2016 Rab8a/Rab11a regulate intercellular communications between neural cells via tunneling nanotubes. Cell death & disease 27 28005071
2014 Rab8 binding to immune cell-specific adaptor LAX facilitates formation of trans-Golgi network-proximal CTLA-4 vesicles for surface expression. Molecular and cellular biology 27 24515439
2019 RAB8A GTPase regulates spindle migration and Golgi apparatus distribution via ROCK-mediated actin assembly in mouse oocyte meiosis†. Biology of reproduction 25 30285101
2018 MEL-pep, an analog of melittin, disrupts cell membranes and reverses 5-fluorouracil resistance in human hepatocellular carcinoma cells. The international journal of biochemistry & cell biology 25 29800725
2017 Disruption of Rab8a and Rab11a causes formation of basolateral microvilli in neonatal enteropathy. Journal of cell science 25 28596241
2004 Mutant presenilin (A260V) affects Rab8 in PC12D cell. Neurochemistry international 25 14643748
2012 EPI64 interacts with Slp1/JFC1 to coordinate Rab8a and Arf6 membrane trafficking. Molecular biology of the cell 24 22219378
2010 Expression and clinicopathological significance of Mel-18 and Bmi-1 mRNA in gastric carcinoma. Journal of experimental & clinical cancer research : CR 23 21059209
2021 Down-regulation of microRNA-30d-5p is associated with gestational diabetes mellitus by targeting RAB8A. Journal of diabetes and its complications 22 34052089
2019 Rab8a localisation and activation by Toll-like receptors on macrophage macropinosomes. Philosophical transactions of the Royal Society of London. Series B, Biological sciences 22 30966999
2016 A novel high-content analysis tool reveals Rab8-driven cytoskeletal reorganization through Rho GTPases, calpain and MT1-MMP. Journal of cell science 22 26940916
2010 Expression of BMI-1 and Mel-18 in breast tissue--a diagnostic marker in patients with breast cancer. BMC cancer 22 21162745
2006 Expression of the melatonin receptor Mel(1c) in neural tissues of the reef fish Siganus guttatus. Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 22 17293145
2017 Endocytic turnover of Rab8 controls cell polarization. Journal of cell science 21 28137756
2005 Ircinin-1 induces cell cycle arrest and apoptosis in SK-MEL-2 human melanoma cells. Molecular carcinogenesis 21 16163705

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