Affinage

RAC1

Ras-related C3 botulinum toxin substrate 1 · UniProt P63000

Audit flag: rerun needed
Length
192 aa
Mass
21.4 kDa
Annotated
2026-04-28
130 papers in source corpus

Mechanistic narrative

Synthesis pass · prose summary of the discoveries below

Parse failed

Mechanism profile

Synthesis pass · controlled-vocabulary classification · explore literature graph →
No controlled-vocabulary terms were assigned to this entry.

Source papers

Stage 0 corpus · 130 papers · ranked by NIH iCite citations
Year Title Journal Citations PMID
1992 The small GTP-binding protein rac regulates growth factor-induced membrane ruffling. Cell 3298 1643658
2004 Mammalian TOR complex 2 controls the actin cytoskeleton and is rapamycin insensitive. Nature cell biology 1726 15467718
2005 A human protein-protein interaction network: a resource for annotating the proteome. Cell 1704 16169070
2002 Generation and initial analysis of more than 15,000 full-length human and mouse cDNA sequences. Proceedings of the National Academy of Sciences of the United States of America 1479 12477932
1994 A brain serine/threonine protein kinase activated by Cdc42 and Rac1. Nature 1377 8107774
2017 Architecture of the human interactome defines protein communities and disease networks. Nature 1085 28514442
2015 A human interactome in three quantitative dimensions organized by stoichiometries and abundances. Cell 1015 26496610
2014 A proteome-scale map of the human interactome network. Cell 977 25416956
2012 Exome sequencing identifies recurrent somatic RAC1 mutations in melanoma. Nature genetics 946 22842228
2009 A genetically encoded photoactivatable Rac controls the motility of living cells. Nature 889 19693014
2020 A reference map of the human binary protein interactome. Nature 849 32296183
2008 Rac activation and inactivation control plasticity of tumor cell movement. Cell 794 18984162
2003 Complete sequencing and characterization of 21,243 full-length human cDNAs. Nature genetics 754 14702039
1996 Wiskott-Aldrich syndrome protein, a novel effector for the GTPase CDC42Hs, is implicated in actin polymerization. Cell 734 8625410
2007 Large-scale mapping of human protein-protein interactions by mass spectrometry. Molecular systems biology 733 17353931
2021 Dual proteome-scale networks reveal cell-specific remodeling of the human interactome. Cell 705 33961781
2012 A census of human soluble protein complexes. Cell 689 22939629
2002 Mechanism of regulation of WAVE1-induced actin nucleation by Rac1 and Nck. Nature 666 12181570
2011 Phylogenetic-based propagation of functional annotations within the Gene Ontology consortium. Briefings in bioinformatics 656 21873635
1998 WAVE, a novel WASP-family protein involved in actin reorganization induced by Rac. The EMBO journal 588 9843499
2000 Localized Rac activation dynamics visualized in living cells. Science (New York, N.Y.) 572 11030651
1995 A conserved binding motif defines numerous candidate target proteins for both Cdc42 and Rac GTPases. The Journal of biological chemistry 552 7493928
1997 Activation of the nuclear factor-kappaB by Rho, CDC42, and Rac-1 proteins. Genes & development 546 9042860
2000 Toll-like receptor 2-mediated NF-kappa B activation requires a Rac1-dependent pathway. Nature immunology 536 11101877
2002 Rac1 and Cdc42 capture microtubules through IQGAP1 and CLIP-170. Cell 502 12110184
2011 Analysis of the myosin-II-responsive focal adhesion proteome reveals a role for β-Pix in negative regulation of focal adhesion maturation. Nature cell biology 490 21423176
2002 Unconventional Rac-GEF activity is mediated through the Dock180-ELMO complex. Nature cell biology 482 12134158
2003 Coactivation of Rac and Rho by Wnt/Frizzled signaling is required for vertebrate gastrulation. Genes & development 470 12533515
1989 rac, a novel ras-related family of proteins that are botulinum toxin substrates. The Journal of biological chemistry 457 2674130
2000 IRSp53 is an essential intermediate between Rac and WAVE in the regulation of membrane ruffling. Nature 454 11130076
2004 Integrins regulate Rac targeting by internalization of membrane domains. Science (New York, N.Y.) 452 14764880
2002 P-Rex1, a PtdIns(3,4,5)P3- and Gbetagamma-regulated guanine-nucleotide exchange factor for Rac. Cell 447 11955434
2003 Hematopoietic cell regulation by Rac1 and Rac2 guanosine triphosphatases. Science (New York, N.Y.) 398 14564009
1997 Requirements for both Rac1 and Cdc42 in membrane ruffling and phagocytosis in leukocytes. The Journal of experimental medicine 341 9348306
2004 Cdc42, Rac1, and Rac2 display distinct patterns of activation during phagocytosis. Molecular biology of the cell 299 15169870
2009 Rac1 GTPase: a "Rac" of all trades. Cellular and molecular life sciences : CMLS 295 19151919
2006 Requirement of Rac1 in the development of cardiac hypertrophy. Proceedings of the National Academy of Sciences of the United States of America 240 16651530
2000 Vav2 is an activator of Cdc42, Rac1, and RhoA. The Journal of biological chemistry 227 10744696
2005 Stem cell depletion through epidermal deletion of Rac1. Science (New York, N.Y.) 215 16081735
1998 Fc receptor-mediated phagocytosis requires CDC42 and Rac1. The EMBO journal 196 9799231
1996 Rac-1 dependent stimulation of the JNK/SAPK signaling pathway by Vav. Oncogene 154 8760286
1998 Characterization of a Rac1- and RhoGDI-associated lipid kinase signaling complex. Molecular and cellular biology 135 9447972
1998 RhoG GTPase controls a pathway that independently activates Rac1 and Cdc42Hs. Molecular biology of the cell 135 9614181
2000 Membrane recruitment of Rac1 triggers phagocytosis. Journal of cell science 120 10934035
1996 The Ras-related GTPase Rac1 binds tubulin. The Journal of biological chemistry 112 8631991
2011 S6K1 and mTOR regulate Rac1-driven platelet activation and aggregation. Blood 111 21757621
2006 Pro-metastatic signaling by c-Met through RAC-1 and reactive oxygen species (ROS). Oncogene 110 16462764
2014 TRPM2 mediates ischemic kidney injury and oxidant stress through RAC1. The Journal of clinical investigation 104 25295536
2007 Rac1 signaling stimulates N-cadherin expression, mesenchymal condensation, and chondrogenesis. The Journal of biological chemistry 104 17573353
2008 cAMP induced Rac 1-mediated cytoskeletal reorganization in microvascular endothelium. Histochemistry and cell biology 91 18392843
2012 CYK4 inhibits Rac1-dependent PAK1 and ARHGEF7 effector pathways during cytokinesis. The Journal of cell biology 90 22945935
2005 Rac1/Cdc42 and RhoA GTPases antagonistically regulate chondrocyte proliferation, hypertrophy, and apoptosis. Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research 90 15883643
2016 Rac1 and RhoA: Networks, loops and bistability. Small GTPases 86 27533896
2009 The small GTPase Rac1 regulates auditory hair cell morphogenesis. The Journal of neuroscience : the official journal of the Society for Neuroscience 83 20016102
2016 Impact of point mutation P29S in RAC1 on tumorigenesis. Tumour biology : the journal of the International Society for Oncodevelopmental Biology and Medicine 81 27699663
2013 miR-320a suppresses colorectal cancer progression by targeting Rac1. Carcinogenesis 80 24265291
2006 Sos-mediated activation of rac1 by p66shc. The Journal of cell biology 78 16520382
2006 E-cadherin engagement stimulates proliferation via Rac1. The Journal of cell biology 78 16682529
2003 Modulation of Rac1 and ARF6 activation during epithelial cell scattering. The Journal of biological chemistry 78 12609992
2021 KDM6A-ARHGDIB axis blocks metastasis of bladder cancer by inhibiting Rac1. Molecular cancer 77 34006303
2010 Focal-adhesion targeting links caveolin-1 to a Rac1-degradation pathway. Journal of cell science 77 20460433
2003 Skeletal muscle signaling pathway through the dystrophin glycoprotein complex and Rac1. The Journal of biological chemistry 76 12885773
2017 Gradients of Rac1 Nanoclusters Support Spatial Patterns of Rac1 Signaling. Cell reports 75 29141223
2018 Compartmentalisation of RAC1 signalling. Current opinion in cell biology 71 29723737
2013 Activation of Rac-1 and RhoA contributes to podocyte injury in chronic kidney disease. PloS one 70 24244677
2020 Sarcoidosis and the mTOR, Rac1, and Autophagy Triad. Trends in immunology 69 32122794
2018 Fam49/CYRI interacts with Rac1 and locally suppresses protrusions. Nature cell biology 69 30250061
2019 Protein prenylation restrains innate immunity by inhibiting Rac1 effector interactions. Nature communications 68 31484924
2016 Differential Rac1 signalling by guanine nucleotide exchange factors implicates FLII in regulating Rac1-driven cell migration. Nature communications 65 26887924
2015 RAC1 P29S regulates PD-L1 expression in melanoma. Pigment cell & melanoma research 63 26176707
2005 Activation of Rac-1 and Cdc42 stabilizes the microvascular endothelial barrier. Histochemistry and cell biology 63 16195887
2002 DOCK2 associates with CrkL and regulates Rac1 in human leukemia cell lines. Blood 63 12393632
2015 Modulation of actin dynamics by Rac1 to target cognitive function. Journal of neurochemistry 61 25818528
2005 Selective Rac-1 inhibition protects from diabetes-induced vascular injury. Circulation research 61 16357302
2018 Optogenetic dissection of Rac1 and Cdc42 gradient shaping. Nature communications 60 30446664
2006 Alsin/Rac1 signaling controls survival and growth of spinal motoneurons. Annals of neurology 59 16802292
2016 Rab7a regulates cell migration through Rac1 and vimentin. Biochimica et biophysica acta. Molecular cell research 57 27888097
2012 Rac1 controls Schwann cell myelination through cAMP and NF2/merlin. The Journal of neuroscience : the official journal of the Society for Neuroscience 56 23197717
2005 Yersinia pseudotuberculosis spatially controls activation and misregulation of host cell Rac1. PLoS pathogens 56 16228016
2008 Beta-PIX and Rac1 GTPase mediate trafficking and negative regulation of NOD2. Journal of immunology (Baltimore, Md. : 1950) 55 18684957
2007 The IQGAP1-Rac1 and IQGAP1-Cdc42 interactions: interfaces differ between the complexes. The Journal of biological chemistry 55 17984089
2004 Regulation of anoikis by Cdc42 and Rac1. Experimental cell research 54 15093747
2004 Diacylglycerol kinase gamma serves as an upstream suppressor of Rac1 and lamellipodium formation. The Journal of biological chemistry 54 15102830
2016 GEFs: Dual regulation of Rac1 signaling. Small GTPases 53 27314616
2012 Serine-71 phosphorylation of Rac1 modulates downstream signaling. PloS one 53 22970203
2018 Post-Translational Modification and Subcellular Distribution of Rac1: An Update. Cells 51 30544910
2014 mTOR regulate EMT through RhoA and Rac1 pathway in prostate cancer. Molecular carcinogenesis 50 25043657
2014 Rac-1 as a new therapeutic target in cerebro- and cardio-vascular diseases. Current drug targets 49 25345393
2006 Rac1 GTPase regulates cell genomic stability and senescence. The Journal of biological chemistry 47 17032649
2019 Transient Activations of Rac1 at the Lamellipodium Tip Trigger Membrane Protrusion. Current biology : CB 46 31422887
2016 Tiam1/Rac1 complex controls Il17a transcription and autoimmunity. Nature communications 46 27725632
2017 Suppression of RAC1-driven malignant melanoma by group A PAK inhibitors. Oncogene 45 29059171
2022 Rac1 as a therapeutic anticancer target: Promises and limitations. Biochemical pharmacology 41 35853497
2007 Reciprocal regulation of Rac1 and Rho1 in Drosophila circulating immune surveillance cells. Journal of cell science 41 17227793
2015 mTOR Directs Breast Morphogenesis through the PKC-alpha-Rac1 Signaling Axis. PLoS genetics 40 26132202
2015 Distinct predictive performance of Rac1 and Cdc42 in cell migration. Scientific reports 40 26634649
2014 Coronin-1C and RCC2 guide mesenchymal migration by trafficking Rac1 and controlling GEF exposure. Journal of cell science 37 25074804
2014 RAC1 and melanoma. Clinical therapeutics 37 25465943
1998 p21ras initiates Rac-1 but not phosphatidyl inositol 3 kinase/PKB, mediated signaling pathways in T lymphocytes. Oncogene 37 9796702
2016 Emerging roles of RAC1 in treating lung cancer patients. Clinical genetics 36 27790713
2014 Rac1 signaling is critical to cardiomyocyte polarity and embryonic heart development. Journal of the American Heart Association 36 25315346
2022 Overexpressed or hyperactivated Rac1 as a target to treat hepatocellular carcinoma. Pharmacological research 35 35405309
2013 GluN3A expression restricts spine maturation via inhibition of GIT1/Rac1 signaling. Proceedings of the National Academy of Sciences of the United States of America 35 24297929
2012 Upon Wnt stimulation, Rac1 activation requires Rac1 and Vav2 binding to p120-catenin. Journal of cell science 34 22946057
2014 CDC-42 and RAC-1 regulate opposite chemotropisms in Neurospora crassa. Journal of cell science 33 24790223
2014 Redox regulation of Rac1 by thiol oxidation. Free radical biology & medicine 33 25289457
2002 Opsonization modulates Rac-1 activation during cell entry by Leishmania amazonensis. Infection and immunity 33 12117970
2013 The small GTPase Rac1 is required for smooth muscle contraction. The Journal of physiology 32 24297853
2019 RHOG Activates RAC1 through CDC42 Leading to Tube Formation in Vascular Endothelial Cells. Cells 31 30781697
2009 Activated Rac1 requires gp130 for Stat3 activation, cell proliferation and migration. Experimental cell research 30 19852956
2002 Participation of small GTPases Rac1 and Cdc42Hs in myoblast transformation. Oncogene 30 11973651
2018 RIT1 controls actin dynamics via complex formation with RAC1/CDC42 and PAK1. PLoS genetics 28 29734338
2005 Regulation of p21-activated kinase-independent Rac1 signal transduction by nischarin. The Journal of biological chemistry 28 16002401
2020 Effect of PAK Inhibition on Cell Mechanics Depends on Rac1. Frontiers in cell and developmental biology 27 32047750
2020 IQGAP1 causes choroidal neovascularization by sustaining VEGFR2-mediated Rac1 activation. Angiogenesis 27 32783108
2018 An Intellectual Disability-Related Missense Mutation in Rac1 Prevents LTP Induction. Frontiers in molecular neuroscience 27 30042656
2009 CCK activates RhoA and Rac1 differentially through Galpha13 and Galphaq in mouse pancreatic acini. American journal of physiology. Cell physiology 26 19940064
2020 Prenylation of Axonally Translated Rac1 Controls NGF-Dependent Axon Growth. Developmental cell 25 32533921
2019 ASIC1a promotes synovial invasion of rheumatoid arthritis via Ca2+/Rac1 pathway. International immunopharmacology 25 31865241
2020 Rac1 Inhibition Via Srgap2 Restrains Inflammatory Osteoclastogenesis and Limits the Clastokine, SLIT3. Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research 24 31880824
2020 Stress-Sensitive Protein Rac1 and Its Involvement in Neurodevelopmental Disorders. Neural plasticity 24 33299404
2013 The N-BAR domain protein, Bin3, regulates Rac1- and Cdc42-dependent processes in myogenesis. Developmental biology 24 23872330
2024 Implication of Rac1 GTPase in molecular and cellular mitochondrial functions. Life sciences 23 38387701
2021 Mechanistic Differences of Activation of Rac1P29S and Rac1A159V. The journal of physical chemistry. B 23 33848152
2017 Discovery and characterization of small molecule Rac1 inhibitors. Oncotarget 23 28410221
2009 Rac1 signaling modulates BCL-6-mediated repression of gene transcription. Molecular and cellular biology 23 19487462
2022 Two Rac1 pools integrate the direction and coordination of collective cell migration. Nature communications 22 36224221
2020 TNFAIP8L2/TIPE2 impairs autolysosome reformation via modulating the RAC1-MTORC1 axis. Autophagy 22 32460619
2018 Verbascoside Attenuates Rac-1 and HIF-1α Signaling Cascade in Colorectal Cancer Cells. Anti-cancer agents in medicinal chemistry 22 29886834
2010 Compromized geranylgeranylation of RhoA and Rac1 in mevalonate kinase deficiency. Journal of inherited metabolic disease 22 20814828