Affinage

DNMBP

Dynamin-binding protein · UniProt Q6XZF7

Length
1577 aa
Mass
177.3 kDa
Annotated
2026-06-09
41 papers in source corpus 13 papers cited in narrative 13 extracted findings
Cross-family judge vs UniProt: Affinage preferred faithfulness: 7/7 claims corpus-supported (100%)

Mechanistic narrative

Synthesis pass · prose summary of the discoveries below

DNMBP (Tuba) is a multidomain scaffold and Cdc42-specific guanine nucleotide exchange factor that couples the membrane-fission machinery to actin regulators and Cdc42 signaling to control epithelial junction geometry, apical polarity, and tissue morphogenesis (PMID:14506234, PMID:17015620). Its four N-terminal SH3 domains bind dynamin with high avidity, a central DH domain selectively activates Cdc42 (not Rac or Rho), an adjacent BAR domain replaces the canonical PH module, and a C-terminal SH3 domain directly engages the actin nucleation-promoting factors N-WASP and Ena/VASP (PMID:14506234, PMID:16413298). At apical cell junctions, DNMBP is recruited through ZO-1 and shapes junctional F-actin and E-cadherin assembly via a Tuba→Cdc42→N-WASP cascade (PMID:17015620). This GEF activity is catalytically required for apical Cdc42 enrichment, which drives aPKC-dependent spindle orientation and single-lumen formation in epithelial cysts, with N-WASP cooperating at the pre-apical patch and a Tuba/Cdc42/Par6A complex restricting Cdc42 to ensure apical domain singularity (PMID:20479467, PMID:21677511, PMID:30408122). The same Tuba→Cdc42 module is deployed for ciliogenesis and nephrogenesis, for DDR1-driven linear invadosome formation and matrix degradation on collagen, and for Rab8a-dependent axon specification and cortical neuronal migration (PMID:25422375, PMID:26895965, PMID:33478991). Under hyperosmotic stress, Nedd4-2 (NEDD4L) ubiquitinates DNMBP and targets it to P-body condensates to enable Cdc42 and downstream p38-MAPK activation (PMID:40975170). Bi-allelic loss-of-function variants in DNMBP cause infantile cataracts in humans, consistent with its role in epithelial junction and E-cadherin regulation (PMID:30290152).

Mechanistic history

Synthesis pass · year-by-year structured walk · 11 steps
  1. 2003 High

    Established the domain architecture and biochemical logic of DNMBP, defining it as a scaffold that physically bridges dynamin to actin regulators while functioning as a Cdc42-specific GEF.

    Evidence Co-IP, pulldowns, in vitro GEF assays, and forced mitochondrial targeting of the C-terminal SH3 domain

    PMID:14506234

    Open questions at the time
    • Cellular context in which dynamin–actin coupling occurs not defined
    • No structural detail of the DH-BAR module
  2. 2005 High

    Confirmed and elaborated the high-avidity dynamin binding by the four SH3 domains and the unusual DH-BAR arrangement, consolidating the Cdc42-specific GEF identity.

    Evidence Biochemical pulldown, co-IP, and GEF activity assays with domain characterization

    PMID:16413298

    Open questions at the time
    • Functional consequence of the BAR domain in lieu of PH not resolved
  3. 2006 High

    Placed DNMBP at apical cell junctions and demonstrated a Tuba→Cdc42→N-WASP pathway shaping junction geometry, F-actin, and E-cadherin, connecting the scaffold to epithelial morphogenesis.

    Evidence RNAi knockdown, calcium-switch junction assays, dominant-active rescue, and ZO-1 co-IP; plus overexpression/knockdown studies of PIP5Kα-driven actin comets and melanoma invasiveness

    PMID:16757518 PMID:17015620

    Open questions at the time
    • Mechanism of ZO-1-mediated apical targeting not fully defined
    • Comet/invasion link is partially indirect
  4. 2010 High

    Demonstrated that DNMBP GEF catalytic activity is required for apical Cdc42 enrichment and correct spindle orientation, establishing Tuba upstream of Cdc42→aPKC in single-lumen morphogenesis.

    Evidence GEF screen, RNAi, rescue with WT vs GEF-dead Tuba and active Cdc42, aPKC activity assay in epithelial cysts

    PMID:20479467

    Open questions at the time
    • How apical Cdc42 spatially couples to spindle machinery not detailed
  5. 2011 Medium

    Showed DNMBP and N-WASP are mutually dependent for pre-apical patch localization, refining the cooperative basis of lumen positioning.

    Evidence RNAi knockdown and multilumen phenotype assays in Caco-2 cysts

    PMID:21677511

    Open questions at the time
    • Functional rescue not fully demonstrated
    • Single lab
  6. 2013 High

    Resolved at atomic resolution how the SH3-6 domain engages N-WASP and Mena and how the Listeria factor InlC competitively hijacks this interface, defining a structural basis for DNMBP's partner binding.

    Evidence Crystal structures of Tuba SH3-6 with InlC, N-WASP and Mena plus F146A mutagenesis and in vivo spreading assays

    PMID:24332715

    Open questions at the time
    • Physiological regulation of SH3-6 occupancy not addressed
  7. 2014 High

    Identified DNMBP as the GEF coupling DDR1 receptor signaling to Cdc42 for linear invadosome formation and collagen degradation, independent of DDR1 kinase activity and Src.

    Evidence siRNA knockdown, Cdc42 activity pulldown, colocalization, and matrix degradation/invasion assays

    PMID:25422375

    Open questions at the time
    • Mechanism by which DDR1 recruits Tuba unknown
  8. 2016 High

    Extended DNMBP function to ciliogenesis and nephrogenesis, showing genetic synergy with Cdc42 across cell and zebrafish models.

    Evidence RNAi in MDCK cells, zebrafish morpholino knockdown, tuba+cdc42 double-morphant synergy, immunofluorescence

    PMID:26895965

    Open questions at the time
    • Molecular link between Tuba and the ciliary apparatus not defined
  9. 2018 High

    Connected DNMBP to human disease and refined a polarity mechanism: LOF variants cause infantile cataracts, and a Tuba/Cdc42/Par6A trimeric complex restricts Cdc42 to ensure apical domain singularity.

    Evidence Exome sequencing with Drosophila sif RNAi and E-cadherin/junction readouts; Co-IP, Par6A CRISPR KO and mutant rescue with live Cdc42 FRAP imaging

    PMID:30290152 PMID:30408122

    Open questions at the time
    • How LOF variants disrupt GEF/scaffold function at molecular level not shown
    • Mechanism of Par6A-mediated Cdc42 spatial restriction incomplete
  10. 2021 High

    Positioned DNMBP downstream of Rab8a in neuronal polarization, identifying a Rab8a→Tuba→Cdc42 axis that specifies axons and drives cortical migration.

    Evidence Gain/loss of function in rat hippocampal neurons, in utero electroporation in mice, immunofluorescence of the Tuba axonal gradient

    PMID:33478991

    Open questions at the time
    • How Rab8a generates the proximal-to-distal Tuba gradient not resolved
  11. 2025 Medium

    Revealed stress-responsive regulation of DNMBP: Nedd4-2 ubiquitinates it and targets it to P-bodies to enable hyperosmotic Cdc42 and p38-MAPK activation.

    Evidence BioID proximity screen, Co-IP, ubiquitination assay, P-body imaging, DNMBP KO and Cdc42/p38 activity assays

    PMID:40975170

    Open questions at the time
    • Not independently replicated
    • Functional consequence of P-body sequestration of DNMBP unclear
    • Role of ubiquitination in GEF activity not defined

Open questions

Synthesis pass · forward-looking unresolved questions
  • How DNMBP's distinct partner interactions (dynamin, N-WASP, ZO-1, Par6A, Rab8a, DDR1, Nedd4-2) are differentially deployed across epithelial, ciliary, neuronal, and stress contexts remains unresolved.
  • No integrated structural model of the full-length protein
  • Determinants of context-specific scaffolding not defined
  • Regulation of GEF output by upstream signals incompletely mapped

Mechanism profile

Synthesis pass · controlled-vocabulary classification · explore literature graph →
Molecular activity
GO:0098772 molecular function regulator activity 4 GO:0060090 molecular adaptor activity 3 GO:0008092 cytoskeletal protein binding 2
Localization
GO:0005856 cytoskeleton 2 GO:0005886 plasma membrane 2 GO:0005929 cilium 1
Pathway
R-HSA-162582 Signal Transduction 4 R-HSA-1266738 Developmental Biology 3 R-HSA-1500931 Cell-Cell communication 2
Complex memberships
Tuba/Cdc42/Par6A trimeric complex

Evidence

Reading pass · 13 per-paper findings extracted from the source corpus
Year Finding Method Journal Conf PMIDs
2003 Tuba (DNMBP) is a scaffold protein containing four N-terminal SH3 domains that bind dynamin, a central DH domain that functions as a Cdc42-specific GEF (not activating Rac or Rho), a BAR domain (which replaces the typical PH domain following DH domains), and a C-terminal SH3 domain that directly binds N-WASP and Ena/VASP proteins, linking dynamin to actin regulatory proteins. Co-immunoprecipitation, pulldown assays, in vitro GEF activity assay, forced mitochondrial targeting of C-terminal SH3 domain to assess F-actin recruitment The Journal of biological chemistry High 14506234
2005 The four N-terminal SH3 domains of Tuba bind dynamin with exceptionally high avidity; the DH domain is a Cdc42-specific GEF unique in being followed by a BAR domain rather than a PH domain; the C-terminal SH3 domain directly binds N-WASP and Ena/VASP and recruits a larger actin regulatory complex. Biochemical pulldown, co-immunoprecipitation, GEF activity assays, domain characterization Methods in enzymology High 16413298
2006 Tuba is concentrated at the apical-most region of cell junctions in simple epithelia via interaction with ZO-1. RNAi-mediated depletion of Tuba alters the geometrical configuration of cell junctions (curved/slack appearance), modifies junctional F-actin and E-cadherin assembly, and retards junction formation. Suppression of Cdc42 or N-WASP mimics Tuba depletion; overexpression of dominant-active Cdc42 or N-WASP rescues Tuba-depleted cells, establishing a Tuba→Cdc42→N-WASP pathway for junction shaping. RNAi knockdown, immunofluorescence, calcium-switch junction formation assay, dominant-active rescue, co-immunoprecipitation with ZO-1 The Journal of cell biology High 17015620
2006 Tuba overexpression stimulates dorsal ruffles and actin-driven motility of intracellular puncta requiring the C-terminal SH3, DH/GEF, and BAR domains. Tuba is recruited to PIP5Kα-generated lipid vesicles and promotes N-WASP-dependent actin comet formation. RNAi knockdown of Tuba attenuates PIP5Kα-generated comet formation and invasive behavior of B16 melanoma cells. Overexpression, RNAi knockdown, fluorescence microscopy, domain deletion analysis, invasiveness assays Journal of cell science Medium 16757518
2010 Tuba, as a Cdc42-specific GEF, is required for Cdc42 enrichment at the apical cortex of epithelial cysts. Loss of Tuba causes a multilumen phenotype by disrupting spindle orientation; this is rescued by human Tuba or constitutively active Cdc42 but not by a GEF-dead Tuba mutant, placing Tuba upstream of Cdc42→aPKC→spindle orientation in epithelial ductal morphogenesis. RNAi screen (70 GEFs), RNAi knockdown, rescue with Tuba WT vs. GEF-dead mutant, active Cdc42 rescue, immunofluorescence, aPKC activity assay The Journal of cell biology High 20479467
2011 Tuba and N-WASP function cooperatively at the pre-apical patch (PAP) to position the central lumen during epithelial cyst morphogenesis; each depends on the other for localization to the PAP, and the cooperative function requires the polyproline region of N-WASP. RNAi knockdown, immunofluorescence localization, multilumen phenotype assay in Caco-2 cysts Cell adhesion & migration Medium 21677511
2013 The Listeria virulence factor InlC binds the sixth SH3 domain (SH3-6) of human Tuba, competitively disrupting its physiological interaction with N-WASP and Mena; the InlC/Tuba SH3-6 interaction is centered on Phe146 of InlC stacking on Asn1569 of Tuba, and replacing Phe146 with Ala largely abrogates affinity and in vivo mimics deletion of inlC. Crystal structure of Tuba SH3-6 complexes with InlC, N-WASP, and Mena; site-directed mutagenesis (F146A); in vivo spreading assays Structure (London, England : 1993) High 24332715
2014 DDR1 (Discoidin Domain Receptor 1) signals through Tuba and Cdc42 to promote linear invadosome formation and matrix degradation on collagen I fibrils; DDR1 kinase activity and Src are not required, but Cdc42 activation by DDR1 is Tuba-dependent, as both Tuba and Cdc42 localize to linear invadosomes and are required for their formation. SiRNA knockdown, immunofluorescence colocalization, Cdc42 activity assay (pulldown), matrix degradation assay, collagen gel invasion assay The Journal of cell biology High 25422375
2016 Tuba (Dynamin Binding Protein) is required for ciliogenesis and nephrogenesis: Tuba knockdown in MDCK cells abolishes primary cilia, impairs apical polarization, and inhibits HGF-induced tubulogenesis. In zebrafish, tuba morphants exhibit ciliary mutant phenotypes in multiple ciliated organs; co-injection of sub-threshold tuba and cdc42 morpholinos causes genetic synergy and disorganized pronephric duct cilia, placing Tuba in the same Cdc42/ciliogenesis pathway. RNAi knockdown in MDCK cells, zebrafish morpholino knockdown, genetic epistasis (tuba + cdc42 double morpholino), immunofluorescence, electroretinography The Journal of biological chemistry High 26895965
2018 Bi-allelic loss-of-function variants in DNMBP cause infantile cataracts in humans. RNAi knockdown of the Drosophila ortholog still life (sif) in lens-secreting cells disrupts lens-secreting cell development, delocalizes E-cadherin, alters septate junction distribution in cone cells, and reduces electroretinography amplitudes. In human epithelial cells, DNMBP regulates tight junction shape and E-cadherin assembly pattern. Exome sequencing (human genetics), Drosophila RNAi knockdown, immunofluorescence (E-cadherin/septate junction localization), electroretinography, human cell knockdown American journal of human genetics High 30290152
2018 A Tuba/Cdc42/Par6A trimeric complex is required to ensure singularity of the apical domain during enterocyte polarization. Tuba, Cdc42, and Par6A co-immunoprecipitate and partially colocalize at the apical membrane; Par6A is required to restrict Cdc42 signaling at the apical domain; rescue experiments using Par6A mutants show that the ability to form this trimeric complex correlates with restoration of apical domain singularity. Co-immunoprecipitation, CRISPR knockout of Par6A, rescue with Par6A mutants, live imaging of active Cdc42 (FRAP), immunofluorescence colocalization PloS one High 30408122
2021 Tuba activates Cdc42 downstream of Rab8a during neuronal polarization. Rab8a activity generates a proximal-to-distal axonal gradient of Tuba in cultured neurons; gain-of-function of Rab8a or Tuba produces supernumerary axons, while loss-of-function abrogates axon specification, phenocopying Cdc42 loss. In vivo, dominant-negative Rab8a or Tuba knockdown impairs cortical neuronal migration in mice. Gain-of-function and loss-of-function (RNAi/dominant negative) in cultured rat hippocampal neurons, in utero electroporation for cortical migration in mice, immunofluorescence of Tuba gradient The Journal of neuroscience High 33478991
2025 The ubiquitin ligase Nedd4-2 (NEDD4L) binds DNMBP/Tuba preferentially under hyperosmotic stress and ubiquitinates it, targeting DNMBP to P-body condensates. DNMBP itself promotes P-body formation under hyperosmolarity. Both Nedd4-2 and DNMBP are required for Cdc42 activation following hyperosmotic treatment; DNMBP knockout suppresses Cdc42 and its downstream effector p38-MAPK. BioID proximity labeling screen (miniTurbo-Nedd4-2), co-immunoprecipitation, ubiquitination assay, P-body localization by immunofluorescence, DNMBP knockout, Cdc42 and p38-MAPK activity assays The Journal of biological chemistry Medium 40975170

Source papers

Stage 0 corpus · 41 papers · ranked by NIH iCite citations
Year Title Journal Citations PMID
2006 Cdc42 GEF Tuba regulates the junctional configuration of simple epithelial cells. The Journal of cell biology 185 17015620
2003 Tuba, a novel protein containing bin/amphiphysin/Rvs and Dbl homology domains, links dynamin to regulation of the actin cytoskeleton. The Journal of biological chemistry 140 14506234
2010 Tuba, a Cdc42 GEF, is required for polarized spindle orientation during epithelial cyst formation. The Journal of cell biology 110 20479467
2014 Discoidin domain receptor 1 controls linear invadosome formation via a Cdc42-Tuba pathway. The Journal of cell biology 93 25422375
2015 Early salpingectomy (TUbectomy) with delayed oophorectomy to improve quality of life as alternative for risk-reducing salpingo-oophorectomy in BRCA1/2 mutation carriers (TUBA study): a prospective non-randomised multicentre study. BMC cancer 90 26286255
2006 Tuba stimulates intracellular N-WASP-dependent actin assembly. Journal of cell science 62 16757518
2023 TUBectomy with delayed oophorectomy as an alternative to risk-reducing salpingo-oophorectomy in high-risk women to assess the safety of prevention: the TUBA-WISP II study protocol. International journal of gynecological cancer : official journal of the International Gynecological Cancer Society 45 37045546
2018 Bi-allelic Loss-of-Function Variants in DNMBP Cause Infantile Cataracts. American journal of human genetics 32 30290152
2021 Deletion of Ulk1 inhibits neointima formation by enhancing KAT2A/GCN5-mediated acetylation of TUBA/α-tubulin in vivo. Autophagy 30 33985412
2019 Autophagic degradation of KAT2A/GCN5 promotes directional migration of vascular smooth muscle cells by reducing TUBA/α-tubulin acetylation. Autophagy 29 31878840
2011 Tuba and N-WASP function cooperatively to position the central lumen during epithelial cyst morphogenesis. Cell adhesion & migration 26 21677511
2005 Tuba, a GEF for CDC42, links dynamin to actin regulatory proteins. Methods in enzymology 26 16413298
2013 Structural details of human tuba recruitment by InlC of Listeria monocytogenes elucidate bacterial cell-cell spreading. Structure (London, England : 1993) 25 24332715
1987 Conditionally lethal tubA alpha-tubulin mutations in Aspergillus nidulans. Molecular & general genetics : MGG 25 3302605
2016 A microalga, Euglena tuba induces apoptosis and suppresses metastasis in human lung and breast carcinoma cells through ROS-mediated regulation of MAPKs. Cancer cell international 22 27366113
2022 DNMBP-AS1 Regulates NHLRC3 Expression by Sponging miR-93-5p/17-5p to Inhibit Colon Cancer Progression. Frontiers in oncology 18 35574307
2016 Dynamin Binding Protein (Tuba) Deficiency Inhibits Ciliogenesis and Nephrogenesis in Vitro and in Vivo. The Journal of biological chemistry 18 26895965
2021 Tuba Activates Cdc42 during Neuronal Polarization Downstream of the Small GTPase Rab8a. The Journal of neuroscience : the official journal of the Society for Neuroscience 8 33478991
2019 Transcriptomic Analysis of Marine Gastropod Hemifusus tuba Provides Novel Insights into Conotoxin Genes. Marine drugs 8 31405144
2014 Phytochemical profile of a microalgae Euglena tuba and its hepatoprotective effect against iron-induced liver damage in Swiss albino mice. Journal of applied microbiology 8 25195957
2008 DNMBP is genetically associated with Alzheimer dementia in the Belgian population. Neurobiology of aging 8 18359537
2005 Sequence diversity of beta-tubulin (tubA) gene in Phaeosphaeria nodorum and P. avenaria. FEMS microbiology letters 8 15972251
2022 Phytochemical Profiling of Microalgae Euglena tuba and Its Anticancer Activity in Dalton's Lymphoma Cells. Frontiers in bioscience (Landmark edition) 7 35468679
2019 TuBA: Tunable biclustering algorithm reveals clinically relevant tumor transcriptional profiles in breast cancer. GigaScience 6 31216036
2007 No association of dynamin binding protein (DNMBP) gene SNPs and Alzheimer's disease. Neurobiology of aging 6 17442457
2023 Selective HDAC6 inhibitor TubA offers neuroprotection after intracerebral hemorrhage via inhibiting neuronal apoptosis. PeerJ 5 37138816
2018 A Tuba/Cdc42/Par6A complex is required to ensure singularity in apical domain formation during enterocyte polarization. PloS one 5 30408122
2019 The first complete mitochondrial genome of Melongenidae from Hemifusus tuba (Neogastropoda: Buccinoidea). Mitochondrial DNA. Part B, Resources 4 33366012
2020 Screening of Ipomoea tuba Leaf Extract for Identification of Bioactive Compounds and Evaluation of Its in vitro Antiproliferative Activity Against MCF-7 and HeLa Cells. Food technology and biotechnology 3 32684790
2020 Euglena tuba extract provides protection against lipopolysaccharide-induced inflammatory response and oxidative stress in mice. Biologia 3 33106705
2017 Tuba-ovarian auto-amputation caused by ovarian teratoma in an adolescent girl. The Turkish journal of pediatrics 3 29168372
2025 Lidocaine could promote the cuproptosis through up-regulating the long noncoding RNA DNMBP-AS1 in Hep-2 cells. BMC cancer 2 39844114
2023 Long non-coding RNA DNMBP-AS1 promotes prostate cancer development by regulating LCLAT1. Systems biology in reproductive medicine 2 36602957
2017 Targeting complete response with upfront bortezomib consolidation versus observation after the achievement of complete response following autologous transplantation for multiple myeloma (TUBA study). Hematological oncology 2 28681529
2009 Association analysis of dynamin-binding protein (DNMBP) on chromosome 10q with late onset Alzheimer's disease in a large caucasian UK sample. American journal of medical genetics. Part B, Neuropsychiatric genetics : the official publication of the International Society of Psychiatric Genetics 2 18452187
2025 DNMBP-AS1/hsa-miR-30a-5p/PGC1α axis suppresses tumor progression of colorectal cancer by inhibiting PKM2-mediated Warburg effect and enhance anti-PD-1 therapy efficacy. Cell death discovery 1 40603870
2025 mPEG-NH2/2-FPBA/TubA exerts anti-hepatocellular carcinoma activity by targeting ABCF1-K430la through the KDM3A-H3K9me2-HIF1A axis. Colloids and surfaces. B, Biointerfaces 1 40663865
2025 The ubiquitin ligase Nedd4-2 promotes localization of DNMBP/Tuba to P-bodies under hyperosmotic stress. The Journal of biological chemistry 1 40975170
2020 A new species of Cnemaspis Strauch 1887 (Squamata: Gekkonidae) from the Langkawi Archipelago, Kedah, Peninsular Malaysia with an updated checklist of the herpetofauna of Tuba Island. Zootaxa 1 33056576
2025 In vitro effects of transient receptor potential channel modulators on human tuba smooth muscle. Advances in medical sciences 0 41197872
2024 In vitro effect of hyoscine-N-butyl bromide and diclofenac sodium in human tuba uterina. Basic & clinical pharmacology & toxicology 0 38803141

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