Affinage

CALU

Calumenin · UniProt O43852

Round 2 refusal Audit flag: rerun needed
Length
315 aa
Mass
37.1 kDa
Annotated
2026-04-28
130 papers in source corpus

Mechanistic narrative

Synthesis pass · prose summary of the discoveries below

No mechanistic findings about CALU (calumenin) in the available literature (corpus is dominated by papers about Calu-1/Calu-3/Calu-6 lung cancer cell lines and large-scale proteomics datasets, none of which describe direct mechanistic experiments on the calumenin protein itself).

Mechanism profile

Synthesis pass · controlled-vocabulary classification · explore literature graph →
No controlled-vocabulary terms were assigned to this entry.

Source papers

Stage 0 corpus · 130 papers · ranked by NIH iCite citations
Year Title Journal Citations PMID
2006 Global, in vivo, and site-specific phosphorylation dynamics in signaling networks. Cell 2861 17081983
2002 Generation and initial analysis of more than 15,000 full-length human and mouse cDNA sequences. Proceedings of the National Academy of Sciences of the United States of America 1479 12477932
2006 A probability-based approach for high-throughput protein phosphorylation analysis and site localization. Nature biotechnology 1336 16964243
2015 The BioPlex Network: A Systematic Exploration of the Human Interactome. Cell 1118 26186194
2017 Architecture of the human interactome defines protein communities and disease networks. Nature 1085 28514442
2015 A human interactome in three quantitative dimensions organized by stoichiometries and abundances. Cell 1015 26496610
2014 A proteome-scale map of the human interactome network. Cell 977 25416956
2018 VIRMA mediates preferential m6A mRNA methylation in 3'UTR and near stop codon and associates with alternative polyadenylation. Cell discovery 829 29507755
2000 DNA cloning using in vitro site-specific recombination. Genome research 815 11076863
2003 Complete sequencing and characterization of 21,243 full-length human cDNAs. Nature genetics 754 14702039
2021 Dual proteome-scale networks reveal cell-specific remodeling of the human interactome. Cell 705 33961781
2012 A census of human soluble protein complexes. Cell 689 22939629
2011 Phylogenetic-based propagation of functional annotations within the Gene Ontology consortium. Briefings in bioinformatics 656 21873635
2011 Global landscape of HIV-human protein complexes. Nature 593 22190034
2017 Anticancer sulfonamides target splicing by inducing RBM39 degradation via recruitment to DCAF15. Science (New York, N.Y.) 533 28302793
2021 Multilevel proteomics reveals host perturbations by SARS-CoV-2 and SARS-CoV. Nature 532 33845483
2006 Hsp90 cochaperone Aha1 downregulation rescues misfolding of CFTR in cystic fibrosis. Cell 517 17110338
2011 Mapping the NPHP-JBTS-MKS protein network reveals ciliopathy disease genes and pathways. Cell 507 21565611
2003 Exploring proteomes and analyzing protein processing by mass spectrometric identification of sorted N-terminal peptides. Nature biotechnology 485 12665801
2004 The status, quality, and expansion of the NIH full-length cDNA project: the Mammalian Gene Collection (MGC). Genome research 438 15489334
2015 A Dynamic Protein Interaction Landscape of the Human Centrosome-Cilium Interface. Cell 433 26638075
2022 OpenCell: Endogenous tagging for the cartography of human cellular organization. Science (New York, N.Y.) 432 35271311
2010 Systematic analysis of human protein complexes identifies chromosome segregation proteins. Science (New York, N.Y.) 421 20360068
2005 Diversification of transcriptional modulation: large-scale identification and characterization of putative alternative promoters of human genes. Genome research 409 16344560
2015 Panorama of ancient metazoan macromolecular complexes. Nature 407 26344197
1983 Structure of the Ki-ras gene of the human lung carcinoma cell line Calu-1. Nature 393 6308465
2021 A proximity-dependent biotinylation map of a human cell. Nature 339 34079125
2014 A quantitative chaperone interaction network reveals the architecture of cellular protein homeostasis pathways. Cell 325 25036637
2006 Culture of Calu-3 cells at the air interface provides a representative model of the airway epithelial barrier. Pharmaceutical research 299 16779708
2006 Association of warfarin dose with genes involved in its action and metabolism. Human genetics 299 17048007
1994 Calu-3: a human airway epithelial cell line that shows cAMP-dependent Cl- secretion. The American journal of physiology 279 7515578
2012 A high-throughput approach for measuring temporal changes in the interactome. Nature methods 273 22863883
2013 The functional interactome landscape of the human histone deacetylase family. Molecular systems biology 235 23752268
1999 Bicarbonate and chloride secretion in Calu-3 human airway epithelial cells. The Journal of general physiology 231 10228185
2000 Characterization of the Calu-3 cell line as a tool to screen pulmonary drug delivery. International journal of pharmaceutics 195 11064206
2002 Permeability characteristics of calu-3 human bronchial epithelial cells: in vitro-in vivo correlation to predict lung absorption in rats. Journal of drug targeting 153 11996084
2008 Release of volatile organic compounds (VOCs) from the lung cancer cell line CALU-1 in vitro. Cancer cell international 143 19025629
2007 Coordinated release of nucleotides and mucin from human airway epithelial Calu-3 cells. The Journal of physiology 140 17656429
1994 CFTR in Calu-3 human airway cells: channel properties and role in cAMP-activated Cl- conductance. The American journal of physiology 139 7515579
2000 Tight junction properties of the immortalized human bronchial epithelial cell lines Calu-3 and 16HBE14o-. The European respiratory journal 133 10885425
2014 The characterization of the human cell line Calu-3 under different culture conditions and its use as an optimized in vitro model to investigate bronchial epithelial function. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 127 25555374
2003 Drug transport and metabolism characteristics of the human airway epithelial cell line Calu-3. Journal of controlled release : official journal of the Controlled Release Society 109 12618029
2013 Metformin impairs glucose consumption and survival in Calu-1 cells by direct inhibition of hexokinase-II. Scientific reports 101 23797762
2010 Cultured human airway epithelial cells (calu-3): a model of human respiratory function, structure, and inflammatory responses. Critical care research and practice 99 20948883
2010 Time- and passage-dependent characteristics of a Calu-3 respiratory epithelial cell model. Drug development and industrial pharmacy 92 20374185
2002 The antiproliferative effect of synthetic peptidyl GH secretagogues in human CALU-1 lung carcinoma cells. Endocrinology 92 11796502
2002 Characterization of basolateral K+ channels underlying anion secretion in the human airway cell line Calu-3. The Journal of physiology 77 11826162
2009 Induction of IL-6 and inhibition of IL-8 secretion in the human airway cell line Calu-3 by urban particulate matter collected with a modified method of PM sampling. Environmental research 76 19304283
1999 Anion selectivity of apical membrane conductance of Calu 3 human airway epithelium. Pflugers Archiv : European journal of physiology 73 10370058
2001 P-glycoprotein efflux pump expression and activity in Calu-3 cells. Journal of pharmaceutical sciences 71 11288109
2008 Arsenic trioxide inhibits the growth of Calu-6 cells via inducing a G2 arrest of the cell cycle and apoptosis accompanied with the depletion of GSH. Cancer letters 70 18539383
2007 In vitro toxicity and permeation of cyclodextrins in Calu-3 cells. Journal of controlled release : official journal of the Controlled Release Society 67 18160169
2001 Multidrug resistance-associated protein-1 functional activity in Calu-3 cells. The Journal of pharmacology and experimental therapeutics 67 11504821
2013 Pharmaceutical applications of the Calu-3 lung epithelia cell line. Expert opinion on drug delivery 65 23730924
2009 P-glycoprotein-mediated transport of moxifloxacin in a Calu-3 lung epithelial cell model. Antimicrobial agents and chemotherapy 63 19188390
1998 Evidence that Calu-3 human airway cells secrete bicarbonate. The American journal of physiology 60 9530182
2002 Oxidant stress stimulates anion secretion from the human airway epithelial cell line Calu-3: implications for cystic fibrosis lung disease. The Journal of physiology 58 12181292
1997 Calcium-stimulated Cl- secretion in Calu-3 human airway cells requires CFTR. The American journal of physiology 58 9435576
2011 YM155, a novel survivin suppressant, enhances taxane-induced apoptosis and tumor regression in a human Calu 6 lung cancer xenograft model. Anti-cancer drugs 57 21389848
2007 2,4-dinitrophenol induces G1 phase arrest and apoptosis in human pulmonary adenocarcinoma Calu-6 cells. Toxicology in vitro : an international journal published in association with BIBRA 50 18276104
2001 Evidence of P-glycoprotein mediated apical to basolateral transport of flunisolide in human broncho-tracheal epithelial cells (Calu-3). British journal of pharmacology 48 11724763
2008 Growth inhibition in antimycin A treated-lung cancer Calu-6 cells via inducing a G1 phase arrest and apoptosis. Lung cancer (Amsterdam, Netherlands) 47 19111365
2001 Modulation of P-glycoprotein activity in Calu-3 cells using steroids and beta-ligands. International journal of pharmaceutics 47 11576779
2012 Evaluation of air-interfaced Calu-3 cell layers for investigation of inhaled drug interactions with organic cation transporters in vitro. International journal of pharmaceutics 45 22265910
2003 Adenosine receptors and phosphodiesterase inhibitors stimulate Cl- secretion in Calu-3 cells. American journal of respiratory cell and molecular biology 44 12714375
2002 Insulin aggregation and asymmetric transport across human bronchial epithelial cell monolayers (Calu-3). Journal of pharmaceutical sciences 44 11948552
1997 Vectorial transcytosis of dimeric IgA by the Calu-3 human lung epithelial cell line: upregulation by IFN-gamma. The American journal of physiology 43 9176261
2017 A Peptide Nucleic Acid against MicroRNA miR-145-5p Enhances the Expression of the Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) in Calu-3 Cells. Molecules (Basel, Switzerland) 41 29286300
2006 Protease-activated receptor regulation of Cl- secretion in Calu-3 cells requires prostaglandin release and CFTR activation. American journal of physiology. Cell physiology 41 16531569
2021 Differential Signaling and Virus Production in Calu-3 Cells and Vero Cells upon SARS-CoV-2 Infection. Biomolecules & therapeutics 39 33504682
2009 Tiron, a ROS scavenger, protects human lung cancer Calu-6 cells against antimycin A-induced cell death. Oncology reports 39 19082470
2008 Pyrogallol inhibits the growth of lung cancer Calu-6 cells via caspase-dependent apoptosis. Chemico-biological interactions 39 19000662
2020 Quantitative estimation of drug permeation through nasal mucosa using in vitro membrane permeability across Calu-3 cell layers for predicting in vivo bioavailability after intranasal administration to rats. European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 38 32057906
2009 Relative contributions of active mediated transport and passive diffusion of fluoroquinolones with various lipophilicities in a Calu-3 lung epithelial cell model. Antimicrobial agents and chemotherapy 38 19822706
1999 PBA increases CFTR expression but at high doses inhibits Cl(-) secretion in Calu-3 airway epithelial cells. The American journal of physiology 36 10516210
1998 Antisense oligonucleotide to PKC-epsilon alters cAMP-dependent stimulation of CFTR in Calu-3 cells. The American journal of physiology 36 9814985
2012 Bicarbonate-dependent chloride transport drives fluid secretion by the human airway epithelial cell line Calu-3. The Journal of physiology 35 22777674
2002 Regulation of intracellular pH in Calu-3 human airway cells. The Journal of physiology 34 11790817
2018 Carbon monoxide releasing molecule-2 suppresses proliferation, migration, invasion, and promotes apoptosis in non-small cell lung cancer Calu-3 cells. European review for medical and pharmacological sciences 33 29687848
2008 Multiple KCNQ potassium channel subtypes mediate basal anion secretion from the human airway epithelial cell line Calu-3. The Journal of membrane biology 33 18264812
2006 Carbopol-mediated paracellular transport enhancement in Calu-3 cell layers. Journal of pharmaceutical sciences 33 16374869
2020 Suitability and functional characterization of two Calu-3 cell models for prediction of drug permeability across the airway epithelial barrier. International journal of pharmaceutics 32 32485216
2020 Comparative toxicity of ultrafine particles around a major airport in human bronchial epithelial (Calu-3) cell model at the air-liquid interface. Toxicology in vitro : an international journal published in association with BIBRA 32 32726611
2009 Identification and functional characterization of breast cancer resistance protein in human bronchial epithelial cells (Calu-3). International journal of pharmaceutics 32 19782742
2005 Two-pore-domain potassium channels support anion secretion from human airway Calu-3 epithelial cells. Pflugers Archiv : European journal of physiology 32 16311719
2004 Dose-dependent effect of FHIT-inducible expression in Calu-1 lung cancer cell line. Oncogene 32 15361849
2017 Evaluation of permeability alteration and epithelial-mesenchymal transition induced by transforming growth factor-β1 in A549, NCI-H441, and Calu-3 cells: Development of an in vitro model of respiratory epithelial cells in idiopathic pulmonary fibrosis. Journal of pharmacological and toxicological methods 31 28259823
2010 Calu-3 cells grown under AIC and LCC conditions: implications for dipeptide uptake and transepithelial transport of substances. European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 31 21195173
2009 Effects of carbonyl cyanide p-(trifluoromethoxy) phenylhydrazone on the growth inhibition in human pulmonary adenocarcinoma Calu-6 cells. Toxicology 31 19819288
2007 Chloride transporting capability of Calu-3 epithelia following persistent knockdown of the cystic fibrosis transmembrane conductance regulator, CFTR. British journal of pharmacology 31 17339840
1999 Human renin mRNA stability is increased in response to cAMP in Calu-6 cells. Hypertension (Dallas, Tex. : 1979) 31 10082506
2022 Applicability of RPMI 2650 and Calu-3 Cell Models for Evaluation of Nasal Formulations. Pharmaceutics 29 35214101
2012 Functional effects of nanoparticle exposure on Calu-3 airway epithelial cells. Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology 27 22415089
2011 Anion secretion by a model epithelium: more lessons from Calu-3. Acta physiologica (Oxford, England) 27 21251238
2009 Eicosanoid release is increased by membrane destabilization and CFTR inhibition in Calu-3 cells. PloS one 27 19847291
2021 The Effect of Allicin on the Proteome of SARS-CoV-2 Infected Calu-3 Cells. Frontiers in microbiology 26 34777295
2006 Altered expression of FANCL confers mitomycin C sensitivity in Calu-6 lung cancer cells. Cancer biology & therapy 26 17106252
2005 Role for protein phosphatase 2A in the regulation of Calu-3 epithelial Na+-K+-2Cl-, type 1 co-transport function. The Journal of biological chemistry 26 15899883
2021 Propagation of SARS-CoV-2 in Calu-3 Cells to Eliminate Mutations in the Furin Cleavage Site of Spike. Viruses 25 34960703
2014 PX-12 induces apoptosis in Calu-6 cells in an oxidative stress-dependent manner. Tumour biology : the journal of the International Society for Oncodevelopmental Biology and Medicine 25 25391429
2013 Establishing a liquid-covered culture of polarized human airway epithelial Calu-3 cells to study host cell response to respiratory pathogens in vitro. Journal of visualized experiments : JoVE 25 23426201
2012 Characterization of Calu-3 cell monolayers as a model of bronchial epithelial transport: organic cation interaction studies. Journal of drug targeting 25 23050869
2000 Properties of CFTR activated by the xanthine derivative X-33 in human airway Calu-3 cells. American journal of physiology. Cell physiology 25 11078708
2014 Bile acids stimulate chloride secretion through CFTR and calcium-activated Cl- channels in Calu-3 airway epithelial cells. American journal of physiology. Lung cellular and molecular physiology 24 24993131
2012 Transport characteristics of clarithromycin, azithromycin and telithromycin, antibiotics applied for treatment of respiratory infections, in Calu-3 cell monolayers as model lung epithelial cells. Die Pharmazie 24 22764569
2002 Transport of HIV-protease inhibitors across 1 alpha,25di-hydroxy vitamin D3-treated Calu-3 cell monolayers: modulation of P-glycoprotein activity. Pharmaceutical research 24 12458676
2018 N-acetyl cysteine reverts the proinflammatory state induced by cigarette smoke extract in lung Calu-3 cells. Redox biology 23 29573703
2001 Antibacterial activity of apical surface fluid from the human airway cell line Calu-3: pharmacologic alteration by corticosteroids and beta(2)-agonists. American journal of respiratory cell and molecular biology 23 11509329
2020 Treatment of human airway epithelial Calu-3 cells with a peptide-nucleic acid (PNA) targeting the microRNA miR-101-3p is associated with increased expression of the cystic fibrosis Transmembrane Conductance Regulator () gene. European journal of medicinal chemistry 22 33127171
2018 Synthesis and evaluation of the cytotoxic activity of Furanaphthoquinones tethered to 1H-1,2,3-triazoles in Caco-2, Calu-3, MDA-MB231 cells. European journal of medicinal chemistry 22 30025347
2012 Basolateral chloride loading by the anion exchanger type 2: role in fluid secretion by the human airway epithelial cell line Calu-3. The Journal of physiology 22 22802585
2012 Dexamethasone regulates CFTR expression in Calu-3 cells with the involvement of chaperones HSP70 and HSP90. PloS one 22 23272037
2001 Differential regulation of Cl- transport proteins by PKC in Calu-3 cells. American journal of physiology. Lung cellular and molecular physiology 22 11238015
2021 Development of an In Vitro Airway Epithelial-Endothelial Cell Culture Model on a Flexible Porous Poly(Trimethylene Carbonate) Membrane Based on Calu-3 Airway Epithelial Cells and Lung Microvascular Endothelial Cells. Membranes 21 33799867
2011 Imbricatolic acid from Juniperus communis L. prevents cell cycle progression in CaLu-6 cells. Planta medica 21 21567359
2008 Pyrogallol inhibits the growth of human lung cancer Calu-6 cells via arresting the cell cycle arrest. Toxicology in vitro : an international journal published in association with BIBRA 21 18652887
2020 Optimization of inhalable liposomal powder formulations and evaluation of their in vitro drug delivery behavior in Calu-3 human lung epithelial cells. International journal of pharmaceutics 20 32593649
2010 The effects of MAPK inhibitors on antimycin A-treated Calu-6 lung cancer cells in relation to cell growth, reactive oxygen species, and glutathione. Molecular and cellular biochemistry 19 19714450
2009 The effect of MAPK inhibitors on arsenic trioxide-treated Calu-6 lung cells in relation to cell death, ROS and GSH levels. Anticancer research 19 19846917
2006 Ambroxol-induced modification of ion transport in human airway Calu-3 epithelia. Biochemical and biophysical research communications 19 16546120
2004 4-Chloro-benzo[F]isoquinoline (CBIQ) activates CFTR chloride channels and KCNN4 potassium channels in Calu-3 human airway epithelial cells. British journal of pharmacology 19 15148241
2022 Differential effect of SARS-CoV-2 infection on stress granule formation in Vero and Calu-3 cells. Frontiers in microbiology 18 36081788
2020 HMGB1-downregulated angulin-1/LSR induces epithelial barrier disruption via claudin-2 and cellular metabolism via AMPK in airway epithelial Calu-3 cells. Biochemical and biophysical research communications 18 32423802
2018 Flos Magnoliae Inhibits Chloride Secretion via ANO1 Inhibition in Calu-3 Cells. The American journal of Chinese medicine 18 29976084
2013 Salbutamol sulfate absorption across Calu-3 bronchial epithelia cell monolayer is inhibited in the presence of common anionic NSAIDs. The Journal of asthma : official journal of the Association for the Care of Asthma 18 23406450
2013 COMMD1 interacts with the COOH terminus of NKCC1 in Calu-3 airway epithelial cells to modulate NKCC1 ubiquitination. American journal of physiology. Cell physiology 18 23515529
2008 Vasoactive intestinal peptide increases cystic fibrosis transmembrane conductance regulator levels in the apical membrane of Calu-3 cells through a protein kinase C-dependent mechanism. The Journal of pharmacology and experimental therapeutics 18 18650246
2006 Identification and membrane localization of electrogenic sodium bicarbonate cotransporters in Calu-3 cells. Biochimica et biophysica acta 18 16857349
2003 Coupling of CFTR-mediated anion secretion to nucleoside transporters and adenosine homeostasis in Calu-3 cells. The Journal of membrane biology 18 12820662
2021 MUC1-C influences cell survival in lung adenocarcinoma Calu-3 cells after SARS-CoV-2 infection. BMB reports 17 33832550